SCHEMBL5329914

SCHEMBL5329914

NC(=O)C(S)N1N=C(C2CCCCC2)c2ccccc2N(c2ccc([N+](=O)[O-])cc2)C1=O

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTH1R Q03431 11/20 0.47
SCN2A Q99250 1/20 0.38
HTT P42858 1/20 0.35
ACHE P22303 1/20 0.34
CCKBR P32239 3/20 0.34
EPHX1 P07099 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5322001 0.82 PTH1R (0.57) PTH1RCCKBR
SCHEMBL5329909 0.80 PTH1R (0.56) PTH1RCCKBR
SCHEMBL5324938 0.77 PTH1R (0.53) PTH1RSCN2AACHECCKBR
SCHEMBL5285139 0.77 PTH1R (0.49) PTH1RCCKBR
SCHEMBL5320334 0.76 PTH1R (0.69) PTH1RSCN2ACCKBRMAPT
SCHEMBL5285921 0.74 SCN2A (0.46) PTH1RSCN2AHTTACHEMAPT
SCHEMBL5323011 0.74 SCN2A (0.46) PTH1RSCN2AHTTACHEMAPT
SCHEMBL5322196 0.73 PTH1R (0.38) PTH1RSCN2AHTTACHEMAPT
SCHEMBL5287349 0.73 PTH1R (0.44) PTH1RHTTCCKBRMAPT
SCHEMBL5328340 0.72 PTH1R (0.50) PTH1RMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129120-A9 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2007-03-22 WO disclosed
WO-2006129120-A2 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2006-12-07 WO disclosed