SCHEMBL5330056

SCHEMBL5330056

Cc1nc(C)c(S(=O)(=O)Nc2ccc(C(=O)O)cc2)s1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.53
TSHR P16473 2/20 0.53
KIT P10721 1/20 0.50
TDP1 Q9NUW8 1/20 0.48
GFER P55789 2/20 0.47
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA9 Q16790 1/20 0.47
RORA P35398 1/20 0.46
RORC P51449 1/20 0.46
RORB Q92753 1/20 0.46
HTT P42858 1/20 0.45
GAA P10253 2/20 0.44
POLB P06746 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CYP26A1 O43174 1/20 0.43
HSD17B13 Q7Z5P4 1/20 0.43
MEN1 O00255 1/20 0.43
NPC1 O15118 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8274518 0.81 HDAC3 (0.60)
SCHEMBL3556136 0.78 RORA (0.60) ALDH1A1TSHRCA12CA1CA2
SCHEMBL25072776 0.75 GAA (0.50) ALDH1A1TSHRTDP1GFERCA12
SCHEMBL25734174 0.72 TDP1 (0.51) ALDH1A1TSHRKITTDP1GFER
SCHEMBL5323420 0.72 GAA (0.58) ALDH1A1TSHRTDP1GFERCA12
SCHEMBL5329438 0.72 ALDH1A1 (0.50) ALDH1A1TSHRTDP1GFERCA12
SCHEMBL3995457 0.71 TAAR1 (0.56) ALDH1A1TSHRKITMEN1KMT2A
SCHEMBL1030477 0.70 GFER (0.83) ALDH1A1TDP1GFERCA12CA1
SCHEMBL25734178 0.69 ALDH1A1 (0.40) ALDH1A1TSHRTDP1GFERHTT
SCHEMBL2959779 0.69 RORA (0.69) RORARORCRORBGAAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007144379-A1 BICYCLIC COMPOUNDS USEFUL AS CATHEPSIN S INBHIBITORS MEDIVIR AB (SE) 2007-12-21 WO disclosed
WO-2007144379-A1 BICYCLIC COMPOUNDS USEFUL AS CATHEPSIN S INBHIBITORS MEDIVIR AB (SE) 2007-12-21 WO disclosed