SCHEMBL5329438

SCHEMBL5329438

Cc1cnc(S(=O)(=O)Nc2ccc(C(=O)O)cc2)s1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
TSHR P16473 2/20 0.50
TDP1 Q9NUW8 1/20 0.48
GFER P55789 2/20 0.47
POLB P06746 1/20 0.47
HSD17B10 Q99714 1/20 0.47
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA9 Q16790 1/20 0.47
MAPK1 P28482 1/20 0.46
HTT P42858 1/20 0.45
GAA P10253 2/20 0.44
CYP26A1 O43174 1/20 0.43
HSD17B13 Q7Z5P4 1/20 0.43
WDR5 P61964 1/20 0.43
TP53 P04637 1/20 0.43
CTSL P07711 1/20 0.43
CTSS P25774 1/20 0.43
CTSK P43235 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25734174 0.75 TDP1 (0.51) ALDH1A1TSHRTDP1GFERPOLB
SCHEMBL5323420 0.75 GAA (0.58) ALDH1A1TSHRTDP1GFERPOLB
SCHEMBL5330056 0.72 ALDH1A1 (0.53) ALDH1A1TSHRTDP1GFERPOLB
SCHEMBL25734215 0.71 TDP1 (0.44) ALDH1A1TSHRTDP1GFERCA12
SCHEMBL1030477 0.70 GFER (0.83) ALDH1A1TDP1GFERPOLBHSD17B10
SCHEMBL5328641 0.69 ALDH1A1 (0.47) ALDH1A1TSHRTDP1GFERPOLB
SCHEMBL25072776 0.69 GAA (0.50) ALDH1A1TSHRTDP1GFERPOLB
SCHEMBL5326508 0.69 ALDH1A1 (0.55) ALDH1A1TSHRTDP1POLBHSD17B10
SCHEMBL25734183 0.69 TDP1 (0.43) ALDH1A1TSHRTDP1GFERPOLB
SCHEMBL5358577 0.69 CTSL (0.46) ALDH1A1TSHRTDP1GFERPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007144379-A1 BICYCLIC COMPOUNDS USEFUL AS CATHEPSIN S INBHIBITORS MEDIVIR AB (SE) 2007-12-21 WO disclosed
WO-2007144379-A1 BICYCLIC COMPOUNDS USEFUL AS CATHEPSIN S INBHIBITORS MEDIVIR AB (SE) 2007-12-21 WO disclosed
WO-2006064286-A1 CATHEPSIN S INHIBITORS MEDIVIR UK LTD (GB) 2006-06-22 WO disclosed