SCHEMBL5330541

SCHEMBL5330541

Cc1ccc2c(c1)NC(=O)N(C1CC(C)(C)CC(C)(C)C1)N=C2C1CCOCC1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTH1R Q03431 3/20 0.37
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
CHRM5 P08912 1/20 0.32
CHRM1 P11229 1/20 0.32
CHRM3 P20309 1/20 0.32
KCNH2 Q12809 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HSD17B10 Q99714 1/20 0.32
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5319865 0.90 PTH1R (0.37) PTH1RCHRM2CHRM4CHRM5CHRM1
SCHEMBL5320857 0.90 PTH1R (0.36) PTH1RCHRM1KDM4EALDH1A1HSD17B10
SCHEMBL5326307 0.84 PTH1R (0.49) PTH1RCHRM2CHRM4CHRM5CHRM1
SCHEMBL5327534 0.83 PTH1R (0.51) PTH1RCHRM2CHRM4CHRM5CHRM1
SCHEMBL5332531 0.82 PTH1R (0.44) PTH1RCHRM2CHRM4CHRM5CHRM1
SCHEMBL5319651 0.80 PTH1R (0.37) PTH1RCHRM1KDM4EALDH1A1HSD17B10
SCHEMBL5323969 0.78 LMNA (0.31) CNR2
SCHEMBL5322785 0.78 CES2 (0.42) PTH1RCHRM1KDM4EALDH1A1HSD17B10
SCHEMBL5331038 0.78 CES2 (0.42) PTH1RCHRM1KDM4EALDH1A1HSD17B10
SCHEMBL5285662 0.78 CES2 (0.42) PTH1RCHRM1KDM4EALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129120-A9 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2007-03-22 WO disclosed
WO-2006129120-A2 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2006-12-07 WO disclosed