SCHEMBL5330899

SCHEMBL5330899

C=CCOC(=O)C(C(C)=O)[C@@H](NC(=O)OC)c1cccc(F)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.49
MAPT P10636 3/20 0.49
CYP2C19 P33261 4/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2D6 P10635 2/20 0.42
ALOX15 P16050 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
TSHR P16473 1/20 0.39
CYP3A4 P08684 1/20 0.39
KDM4E B2RXH2 1/20 0.37
CNR2 P34972 1/20 0.36
HDAC4 P56524 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC5 Q9UQL6 1/20 0.35
MTOR P42345 1/20 0.35
POLB P06746 1/20 0.34
MAPK1 P28482 1/20 0.34
LMNA P02545 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5330894 1.00 ALDH1A1 (0.49) ALDH1A1MAPTCYP2C19CYP2C9CYP2D6
SCHEMBL14624818 0.88 ALDH1A1 (0.45) ALDH1A1MAPTCYP2C19CYP2C9CYP2D6
SCHEMBL5308650 0.86 ALDH1A1 (0.50) ALDH1A1MAPTCYP2C19CYP2C9CYP2D6
SCHEMBL5308646 0.86 ALDH1A1 (0.50) ALDH1A1MAPTCYP2C19CYP2C9CYP2D6
SCHEMBL14625121 0.86 ALDH1A1 (0.45) ALDH1A1MAPTCYP2C19CYP2C9CYP2D6
SCHEMBL14625355 0.86 CYP3A4 (0.52) ALDH1A1MAPTCYP2C19CYP2C9CYP2D6
SCHEMBL14625468 0.86 CYP2C19 (0.48) ALDH1A1MAPTCYP2C19CYP2C9CYP2D6
SCHEMBL5307157 0.83 MAPT (0.49) ALDH1A1MAPTCYP2C19CYP2C9CYP2D6
SCHEMBL5307158 0.83 MAPT (0.49) ALDH1A1MAPTCYP2C19CYP2C9CYP2D6
SCHEMBL14625714 0.82 MAPT (0.48) ALDH1A1MAPTCYP2C19CYP2D6MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007011910-A2 CHIRAL AMINE-CATALYZED ASYMMETRIC ADDITION OF CARBON-CENTERED NUCLEOPHILES TO IMINES TRUSTEES OF BOSTON UNIVERSITY (US) 2007-01-25 WO disclosed
WO-2007011910-A2 CHIRAL AMINE-CATALYZED ASYMMETRIC ADDITION OF CARBON-CENTERED NUCLEOPHILES TO IMINES TRUSTEES OF BOSTON UNIVERSITY (US) 2007-01-25 WO disclosed