SCHEMBL5308646

SCHEMBL5308646

C=CCOC(=O)C(C(C)=O)C(NC(=O)OC)c1ccc(F)cc1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.50
MAPT P10636 5/20 0.50
CYP3A4 P08684 2/20 0.40
CYP2C19 P33261 2/20 0.40
TSHR P16473 3/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2D6 P10635 1/20 0.38
HTT P42858 2/20 0.33
GRM2 Q14416 1/20 0.33
GRM3 Q14832 1/20 0.33
NOS3 P29474 3/20 0.33
NOS1 P29475 3/20 0.33
NOS2 P35228 3/20 0.33
SLC6A9 P48067 1/20 0.32
SLC6A5 Q9Y345 1/20 0.32
FAAH O00519 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5308650 1.00 ALDH1A1 (0.50) ALDH1A1MAPTCYP3A4CYP2C19TSHR
SCHEMBL14625355 0.88 CYP3A4 (0.52) ALDH1A1MAPTCYP3A4CYP2C19CYP2C9
SCHEMBL5330894 0.86 ALDH1A1 (0.49) ALDH1A1MAPTCYP3A4CYP2C19TSHR
SCHEMBL5330899 0.86 ALDH1A1 (0.49) ALDH1A1MAPTCYP3A4CYP2C19TSHR
SCHEMBL14625714 0.84 MAPT (0.48) ALDH1A1MAPTCYP3A4CYP2C19TSHR
SCHEMBL5307157 0.82 MAPT (0.49) ALDH1A1MAPTCYP3A4CYP2C19TSHR
SCHEMBL5307158 0.82 MAPT (0.49) ALDH1A1MAPTCYP3A4CYP2C19TSHR
SCHEMBL14624818 0.81 ALDH1A1 (0.45) ALDH1A1MAPTCYP3A4CYP2C19TSHR
SCHEMBL14625121 0.79 ALDH1A1 (0.45) ALDH1A1MAPTCYP3A4CYP2C19TSHR
SCHEMBL5325384 0.79 POLB (0.39) ALDH1A1MAPTCYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007011910-A2 CHIRAL AMINE-CATALYZED ASYMMETRIC ADDITION OF CARBON-CENTERED NUCLEOPHILES TO IMINES TRUSTEES OF BOSTON UNIVERSITY (US) 2007-01-25 WO disclosed