SCHEMBL5332052

SCHEMBL5332052

O=C(CSc1nnc(Cc2ccc3c(c2)OCO3)n1-c1ccccc1)NN=Cc1ccco1

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.58
TP53 P04637 1/20 0.57
ALDH1A1 P00352 11/20 0.55
LMNA P02545 1/20 0.55
MAPT P10636 1/20 0.55
NPSR1 Q6W5P4 3/20 0.51
HTT P42858 3/20 0.51
KDM4E B2RXH2 2/20 0.51
RECQL P46063 1/20 0.50
TSHR P16473 2/20 0.49
KMT2A Q03164 2/20 0.49
MAPK1 P28482 2/20 0.49
CYP3A4 P08684 2/20 0.49
CYP2D6 P10635 2/20 0.49
USP2 O75604 1/20 0.48
CYP1A2 P05177 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
NPC1 O15118 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5332046 1.00 POLB (0.58) POLBTP53ALDH1A1LMNAMAPT
SCHEMBL5331032 0.90 POLB (0.62) POLBALDH1A1NPSR1HTTKDM4E
SCHEMBL5331037 0.90 POLB (0.62) POLBALDH1A1NPSR1HTTKDM4E
SCHEMBL5330386 0.88 TP53 (0.67) POLBTP53ALDH1A1LMNAMAPT
SCHEMBL5330392 0.88 TP53 (0.67) POLBTP53ALDH1A1LMNAMAPT
SCHEMBL14542416 0.87 TP53 (0.69) POLBTP53ALDH1A1LMNAMAPT
SCHEMBL5333044 0.84 ALDH1A1 (0.58) POLBTP53ALDH1A1LMNAMAPT
SCHEMBL5333050 0.84 ALDH1A1 (0.58) POLBTP53ALDH1A1LMNAMAPT
SCHEMBL5332252 0.84 POLB (0.68) POLBALDH1A1NPSR1HTTKDM4E
SCHEMBL14542263 0.79 ALDH1A1 (0.69) POLBTP53ALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007047394-A2 THIOTRIAZOLYL DERIVATIVES EPIX DELAWARE, INC. (US) 2007-04-26 WO claimed
WO-2007047394-A2 THIOTRIAZOLYL DERIVATIVES EPIX DELAWARE, INC. (US) 2007-04-26 WO disclosed