SCHEMBL5332533

SCHEMBL5332533

FC(F)(F)c1cccc(-c2cc(Cl)n3ncnc3n2)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.62
KDM4E B2RXH2 8/20 0.62
TP53 P04637 1/20 0.59
HPGD P15428 3/20 0.59
POLB P06746 1/20 0.59
SMN1; SMN2 Q16637 4/20 0.47
TSHR P16473 4/20 0.47
MAPT P10636 2/20 0.47
HTT P42858 2/20 0.47
NPSR1 Q6W5P4 2/20 0.47
USP2 O75604 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
HSD17B10 Q99714 1/20 0.47
GAA P10253 3/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
KDM1A O60341 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11483564 0.85 KDM4E (0.62) ALDH1A1KDM4ETP53HPGDPOLB
SCHEMBL5327134 0.83 ALDH1A1 (0.50) ALDH1A1KDM4ETP53HPGDPOLB
SCHEMBL8124409 0.79 KDM4E (0.51) ALDH1A1KDM4ETP53HPGDPOLB
SCHEMBL11472275 0.78 KCNN3 (0.50) ALDH1A1KDM4ETP53HPGDCYP1A2
SCHEMBL11478689 0.76 KDM4E (1.00) ALDH1A1KDM4ETP53HPGDPOLB
SCHEMBL12953521 0.75 CDK2 (0.48) ALDH1A1KDM4ETP53HPGDSMN1; SMN2
SCHEMBL13304976 0.75 IDO1 (0.42) ALDH1A1KDM4EHPGDSMN1; SMN2TSHR
SCHEMBL14626100 0.74 KDM4E (0.50) ALDH1A1KDM4ETP53HPGDPOLB
SCHEMBL5329221 0.74 KDM4E (0.49) ALDH1A1KDM4ETP53HPGDPOLB
SCHEMBL14626235 0.74 KDM4E (0.49) ALDH1A1KDM4ETP53HPGDPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007011759-A2 INHIBITORS OF MITOTIC KINESIN KALYPSYS, INC. (US) 2007-01-25 WO disclosed
US-4209621-A TRANQUILIZERS AMERICAN CYANAMID COMPANY (US) 1980-06-24 US disclosed