SCHEMBL8124409

SCHEMBL8124409

FC(F)(F)c1cccc(-c2c(Cl)nc3ncnn3c2Cl)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.51
ALDH1A1 P00352 8/20 0.51
HPGD P15428 4/20 0.48
POLB P06746 1/20 0.48
TP53 P04637 1/20 0.46
MBOAT4 Q96T53 2/20 0.45
TSHR P16473 4/20 0.44
SMN1; SMN2 Q16637 4/20 0.44
GAA P10253 3/20 0.44
HTT P42858 3/20 0.44
NPSR1 Q6W5P4 3/20 0.44
MAPT P10636 3/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
CCNA2 P20248 1/20 0.42
CDK2 P24941 1/20 0.42
CDK5 Q00535 1/20 0.42
DYRK1A Q13627 1/20 0.42
CDK5R1 Q15078 1/20 0.42
DYRK2 Q92630 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8117570 0.83 EGLN2 (0.48) KDM4EALDH1A1HPGDPOLBTP53
SCHEMBL8126098 0.83 EGLN2 (0.50) KDM4EALDH1A1HPGDPOLBTSHR
SCHEMBL8124326 0.81 TP53 (0.52) KDM4EALDH1A1HPGDPOLBTP53
SCHEMBL868326 0.80 KDM4E (0.49) KDM4EALDH1A1HPGDPOLBTSHR
SCHEMBL6806818 0.79 MBOAT4 (0.45) KDM4EALDH1A1HPGDPOLBTP53
SCHEMBL5332533 0.79 ALDH1A1 (0.62) KDM4EALDH1A1HPGDPOLBTP53
SCHEMBL8127316 0.78 EGLN2 (0.51) KDM4EALDH1A1HPGDTP53TSHR
SCHEMBL8117996 0.77 KDM4E (0.47) KDM4EALDH1A1HPGDPOLBTSHR
SCHEMBL4820351 0.77 TSHR (0.45) KDM4EALDH1A1HPGDPOLBTP53
SCHEMBL8117510 0.76 KDM4E (0.54) KDM4EALDH1A1HPGDPOLBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0782997-B1 Triazolopyrimidine derivatives SHELL INT RESEARCH (NL) 2000-04-26 EP claimed
EP-0782997-A2 Triazolopyrimidine derivatives SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1997-07-09 EP claimed
EP-0999856-A2 RADIOPHARMACEUTICALS FOR IMAGING INFECTION AND INFLAMMATION Du Pont Pharmaceuticals Company (US) 2000-05-17 EP disclosed
EP-0782997-B1 Triazolopyrimidine derivatives SHELL INT RESEARCH (NL) 2000-04-26 EP disclosed
WO-1998015295-A2 RADIOPHARMACEUTICALS FOR IMAGING INFECTION AND INFLAMMATION DUPONT PHARMACEUTICALS COMPANY (US) 1998-04-16 WO disclosed