SCHEMBL5333831

SCHEMBL5333831

Cc1nc(Nc2ccccc2)sc1S(=O)(=O)N1CCN(C)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
GAA P10253 2/20 0.49
POLB P06746 3/20 0.47
ADORA3 P0DMS8 1/20 0.46
ADORA2A P29274 1/20 0.46
CDK4 P11802 3/20 0.46
CCND1 P24385 3/20 0.46
CDK6 Q00534 3/20 0.46
CCNT1 O60563 3/20 0.46
CDK9 P50750 3/20 0.46
CDK11A Q9UQ88 2/20 0.46
NPC1 O15118 5/20 0.46
RAB9A P51151 5/20 0.46
MAPT P10636 5/20 0.46
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
TP53 P04637 2/20 0.46
LMNA P02545 1/20 0.46
NFKB1 P19838 1/20 0.46
NFKB2 Q00653 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL998661 0.72 MMP1 (0.43) POLBMAPTMEN1KMT2ACA12
SCHEMBL1939520 0.70 MAPT (0.38) ALDH1A1POLBCDK4CCND1CDK6
SCHEMBL999510 0.68 PDE7A (0.40) ALDH1A1NPC1RAB9AKMT2AHPGD
SCHEMBL3936569 0.66 POLB (1.00) ALDH1A1GAAPOLBMEN1KMT2A
SCHEMBL9666910 0.65 MAPT (0.52) ALDH1A1GAAPOLBADORA3ADORA2A
SCHEMBL18711331 0.65 LPAR2 (0.49) ALDH1A1GAAPOLBMEN1KMT2A
SCHEMBL25804386 0.65 ALDH1A1 (0.69) ALDH1A1GAAPOLBNPC1RAB9A
SCHEMBL4001428 0.65 POLB (0.56) ALDH1A1POLBKMT2ALMNASMN1; SMN2
SCHEMBL4765972 0.65 NPC1 (0.76) ALDH1A1GAAPOLBNPC1RAB9A
SCHEMBL4400357 0.65 RAB9A (0.86) ALDH1A1GAAPOLBADORA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1851225-A1 PYRAZOLO-PYRIMIDINE DERIVATIVES AS MGLUR2 ANTAGONISTS F. Hoffmann-Roche AG (CH) 2007-11-07 EP disclosed
WO-2006084634-A1 PYRAZOLO-PYRIMIDINE DERIVATIVES AS MGLUR2 ANTAGONISTS F.HOFFMANN-LA ROCHE AG (CH) 2006-08-17 WO disclosed