SCHEMBL5334834

SCHEMBL5334834

COc1cc2c(cc1OC)C(C)N(C(=O)N1c3ccccc3Sc3ccccc31)CC2

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.59
NPC1 O15118 2/20 0.58
POLB P06746 1/20 0.58
ALDH1A1 P00352 3/20 0.54
TRPV1 Q8NER1 1/20 0.54
KMT2A Q03164 5/20 0.53
HTT P42858 5/20 0.53
GAA P10253 2/20 0.53
TSHR P16473 1/20 0.53
RAB9A P51151 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
MAPT P10636 2/20 0.53
LMNA P02545 2/20 0.51
MAPK1 P28482 1/20 0.51
NCOA1 Q15788 1/20 0.50
NCOA3 Q9Y6Q9 1/20 0.50
MEN1 O00255 1/20 0.50
HPGD P15428 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5243083 0.82 KMT2A (0.49) SMN1; SMN2NPC1POLBALDH1A1KMT2A
SCHEMBL5240550 0.78 ALDH1A1 (0.59) SMN1; SMN2NPC1POLBALDH1A1TRPV1
SCHEMBL5280780 0.77 BCHE (0.52) ALDH1A1KMT2ATSHRMAPTLMNA
SCHEMBL5241937 0.76 BCHE (0.44) SMN1; SMN2NPC1POLBALDH1A1KMT2A
SCHEMBL5350976 0.75 KMT2A (0.55) ALDH1A1KMT2AHTTGAATSHR
SCHEMBL1219345 0.72 HTT (0.66) SMN1; SMN2NPC1POLBALDH1A1KMT2A
SCHEMBL9509837 0.71 SMN1; SMN2 (0.71) SMN1; SMN2NPC1POLBALDH1A1KMT2A
SCHEMBL22970639 0.71 SMN1; SMN2 (0.71) SMN1; SMN2NPC1POLBALDH1A1KMT2A
SCHEMBL5466400 0.71 ALDH1A1 (0.56) SMN1; SMN2POLBALDH1A1KMT2ATSHR
SCHEMBL1219835 0.70 SMN1; SMN2 (0.72) SMN1; SMN2NPC1POLBALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1833797-A1 AZACYCLIC COMPOUNDS AS INHBITORS OF SENSORY NEURONE SPECIFIC CHANNELS (SNS) VERNALIS (R&D) LTD (GB) 2007-09-19 EP disclosed
WO-2006082354-A1 AZACYCLIC COMPOUNDS AS INHIBITORS OF SENSORY NEURONE SPECIFIC CHANNELS ( SNS ) VERNALIS (R & D) LIMITED (GB) 2006-08-10 WO disclosed