SCHEMBL5335903

SCHEMBL5335903

O=C(O)CSc1nnc(-c2cccnc2)n1C1CCCCC1

nearest known ligand 0.76

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HPGD P15428 5/20 0.76
KMT2A Q03164 3/20 0.76
MEN1 O00255 2/20 0.76
MDM2 Q00987 1/20 0.76
GAA P10253 1/20 0.76
ALDH1A1 P00352 4/20 0.72
TSHR P16473 2/20 0.60
NTRK1 P04629 1/20 0.54
NTRK2 Q16620 1/20 0.54
KDM4E B2RXH2 2/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
RXFP1 Q9HBX9 1/20 0.53
ADRB2 P07550 1/20 0.52
RAB9A P51151 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5336800 0.88 KMT2A (0.80) HPGDKMT2AMEN1MDM2GAA
SCHEMBL18559068 0.87 HPGD (1.00) HPGDKMT2AMEN1MDM2GAA
SCHEMBL18559069 0.87 HPGD (1.00) HPGDKMT2AMEN1MDM2GAA
SCHEMBL18556574 0.84 HPGD (1.00) HPGDKMT2AMEN1MDM2GAA
SCHEMBL18556573 0.83 HPGD (1.00) HPGDKMT2AMEN1MDM2GAA
SCHEMBL18556575 0.82 HPGD (1.00) HPGDKMT2AMEN1MDM2GAA
SCHEMBL5327274 0.82 GAA (0.79) HPGDKMT2AMEN1MDM2GAA
SCHEMBL13831971 0.81 TSHR (0.72) HPGDKMT2AMEN1MDM2GAA
SCHEMBL14542264 0.78 HPGD (0.65) HPGDKMT2AMEN1MDM2GAA
SCHEMBL5480773 0.78 ALDH1A1 (0.78) GAAALDH1A1TSHRKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007047394-A2 THIOTRIAZOLYL DERIVATIVES EPIX DELAWARE, INC. (US) 2007-04-26 WO disclosed