SCHEMBL5337615

SCHEMBL5337615

Cc1csc(-c2c(C)ccn2-c2ccc(S(N)(=O)=O)cc2)c1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.40
PTGS1 P23219 11/20 0.40
CA2 P00918 3/20 0.39
CA12 O43570 2/20 0.39
CA1 P00915 2/20 0.39
CA9 Q16790 2/20 0.39
CA3 P07451 1/20 0.39
CA6 P23280 1/20 0.39
CA5A P35218 1/20 0.39
CA7 P43166 1/20 0.39
CA5B Q9Y2D0 1/20 0.39
GHSR Q92847 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL348734 0.80 PTGS2 (0.44) PTGS2PTGS1CA2CA12CA1
SCHEMBL7216201 0.80 PTGS2 (0.52) PTGS2PTGS1CA2CA12CA1
SCHEMBL3690377 0.77 PTGS2 (0.41) PTGS2PTGS1CA2CA12CA1
SCHEMBL2465658 0.77 PTGS2 (0.60) PTGS2PTGS1CA2CA12CA1
SCHEMBL5333903 0.72 PTGS2 (0.60) PTGS2PTGS1CA2CA12CA1
SCHEMBL3690374 0.70 PTGS2 (0.47) PTGS2PTGS1CA2CA12CA1
SCHEMBL5337610 0.70 PTGS2 (0.47) PTGS2PTGS1CA2CA12CA1
SCHEMBL5309164 0.70 CA1 (0.55) PTGS2PTGS1CA2CA12CA1
SCHEMBL27448843 0.70 CA2 (0.53) PTGS2PTGS1CA2CA12CA1
SCHEMBL8121686 0.70 CYP2C9 (0.55) PTGS2PTGS1CA2CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0799823-B1 1,2-Diphenylpyrrole derivatives, their preparation and their therapeutic uses DAIICHI SANKYO CO LTD (JP) 2007-10-31 EP disclosed
US-RE39420-E1 1,2-Diphenylpyrrole derivatives, their preparation and their therapeutic uses SANKYO COMPANY, LIMITED (JP) 2006-12-05 US disclosed
US-5908858-A OSTEOPOROSIS; LEUKOTRIENE INHIBITOR SANKYO COMPANY, LIMITED (JP) 1999-06-01 US disclosed
EP-0799823-A1 1,2-Diphenylpyrrole derivatives, their preparation and their therapeutic uses SANKYO COMPANY LIMITED (JP) 1997-10-08 EP disclosed