SCHEMBL533824

SCHEMBL533824

O=C(O)N1CC[C@](O)(c2ccc(F)c(F)c2)[C@@H](c2onc(-c3ccccc3Cl)c2Br)C1

nearest known ligand 0.67

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
REN P00797 14/20 0.67
KCNH2 Q12809 13/20 0.67
CYP3A4 P08684 12/20 0.67
RAB9A P51151 1/20 0.40
NR1H4 Q96RI1 2/20 0.35
ALDH1A1 P00352 2/20 0.35
NPC1 O15118 1/20 0.35
TSHR P16473 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL555815 0.89 REN (0.61) RENKCNH2CYP3A4RAB9A
SCHEMBL3719090 0.87 REN (0.68) RENKCNH2CYP3A4
SCHEMBL533832 0.84 REN (0.54) RENKCNH2CYP3A4NR1H4
SCHEMBL555742 0.83 REN (0.62) RENKCNH2CYP3A4
SCHEMBL557187 0.80 REN (1.00) RENKCNH2CYP3A4
SCHEMBL555816 0.80 REN (0.56) RENKCNH2CYP3A4RAB9ANR1H4
SCHEMBL557036 0.80 REN (0.60) RENKCNH2CYP3A4NR1H4
SCHEMBL556026 0.79 REN (0.56) RENKCNH2CYP3A4
SCHEMBL557228 0.78 REN (0.53) RENKCNH2CYP3A4
SCHEMBL556767 0.78 REN (0.48) RENKCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2413941-A1 RENIN INHIBITORS Merck Sharp & Dohme Corp. (US) 2012-02-08 EP disclosed
WO-2010114978-A1 RENIN INHIBITORS MERCK SHARP & DOHME CORP. (US) 2010-10-07 WO disclosed