SCHEMBL3719090

SCHEMBL3719090

Cc1cccc(-c2noc(C3CN(C(=O)O)CCC3(O)c3ccc(F)c(F)c3)c2Br)c1C

nearest known ligand 0.68

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
REN P00797 17/20 0.68
KCNH2 Q12809 16/20 0.68
CYP3A4 P08684 13/20 0.68
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
OPRK1 P41145 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL555594 0.90 REN (0.63) RENKCNH2CYP3A4
SCHEMBL533844 0.90 REN (0.63) RENKCNH2CYP3A4
SCHEMBL533824 0.87 REN (0.67) RENKCNH2CYP3A4
SCHEMBL533832 0.83 REN (0.54) RENKCNH2CYP3A4
SCHEMBL555595 0.82 REN (0.58) RENKCNH2CYP3A4
SCHEMBL557568 0.81 REN (1.00) RENKCNH2CYP3A4
SCHEMBL555742 0.78 REN (0.62) RENKCNH2CYP3A4
SCHEMBL555657 0.78 REN (0.62) RENKCNH2CYP3A4
SCHEMBL555815 0.78 REN (0.61) RENKCNH2CYP3A4
SCHEMBL556767 0.77 REN (0.48) RENKCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010114978-A1 RENIN INHIBITORS MERCK SHARP & DOHME CORP. (US) 2010-10-07 WO disclosed