SCHEMBL533832

SCHEMBL533832

Cc1ccc(Cl)c(-c2noc([C@H]3CN(C(=O)O)CC[C@]3(O)c3ccc(F)c(F)c3)c2Br)c1F

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
REN P00797 13/20 0.54
KCNH2 Q12809 12/20 0.54
CYP3A4 P08684 11/20 0.54
NR1H4 Q96RI1 6/20 0.33
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL557210 0.90 REN (0.50) RENKCNH2CYP3A4NR1H4KMT2A
SCHEMBL533824 0.84 REN (0.67) RENKCNH2CYP3A4NR1H4
SCHEMBL3719090 0.83 REN (0.68) RENKCNH2CYP3A4
SCHEMBL557211 0.82 REN (0.46) RENKCNH2CYP3A4NR1H4
SCHEMBL556389 0.82 REN (0.80) RENKCNH2CYP3A4
SCHEMBL557036 0.80 REN (0.60) RENKCNH2CYP3A4NR1H4
SCHEMBL555815 0.75 REN (0.61) RENKCNH2CYP3A4
SCHEMBL555742 0.74 REN (0.62) RENKCNH2CYP3A4
SCHEMBL555594 0.73 REN (0.63) RENKCNH2CYP3A4KMT2A
SCHEMBL533844 0.73 REN (0.63) RENKCNH2CYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2413941-A1 RENIN INHIBITORS Merck Sharp & Dohme Corp. (US) 2012-02-08 EP disclosed
WO-2010114978-A1 RENIN INHIBITORS MERCK SHARP & DOHME CORP. (US) 2010-10-07 WO disclosed