SCHEMBL533862

SCHEMBL533862

Cc1cc(Br)ccc1[C@H]1CNCC[C@@H]1c1cccnc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
REN P00797 2/20 0.45
KCNH2 Q12809 1/20 0.45
KDM1A O60341 1/20 0.42
CHRNB2 P17787 6/20 0.40
CHRNA4 P43681 6/20 0.40
CHRNA7 P36544 3/20 0.37
CYP2A6 P11509 3/20 0.37
MEN1 O00255 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C19 P33261 2/20 0.36
KMT2A Q03164 2/20 0.36
POLB P06746 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CHRNB4 P30926 2/20 0.34
CHRNA3 P32297 2/20 0.34
MAPT P10636 1/20 0.34
TSHR P16473 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL533861 1.00 REN (0.45) RENKCNH2KDM1ACHRNB2CHRNA4
SCHEMBL533991 0.86 REN (0.54) RENKCNH2KDM1ACHRNB2CHRNA4
SCHEMBL534491 0.74 SPR (0.37) CHRNB2CHRNA4CHRNA7MAPTTSHR
SCHEMBL7869555 0.73 REN (0.49) RENKCNH2KDM1A
SCHEMBL10202445 0.73 REN (0.60) RENKCNH2KDM1A
SCHEMBL16271996 0.73 KDM1A (0.52) KDM1ACHRNB2CHRNA4CHRNA7CYP2A6
SCHEMBL10202449 0.72 REN (0.85) RENKCNH2
SCHEMBL555694 0.72 REN (0.85) RENKCNH2
SCHEMBL534462 0.72 MAPT (0.40) CYP2A6MEN1CYP2C19KMT2APOLB
SCHEMBL555812 0.72 MAPT (0.40) CYP2A6MEN1CYP2C19KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2413941-A1 RENIN INHIBITORS Merck Sharp & Dohme Corp. (US) 2012-02-08 EP disclosed
WO-2010114978-A1 RENIN INHIBITORS MERCK SHARP & DOHME CORP. (US) 2010-10-07 WO disclosed