SCHEMBL533991

SCHEMBL533991

Clc1cc(Br)ccc1[C@H]1CNCC[C@@H]1c1cccnc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
REN P00797 2/20 0.54
KCNH2 Q12809 2/20 0.54
KDM1A O60341 1/20 0.42
CHRNB2 P17787 6/20 0.40
CHRNA4 P43681 6/20 0.40
CHRNA7 P36544 2/20 0.37
CYP2A6 P11509 2/20 0.37
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C19 P33261 2/20 0.36
POLB P06746 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
ROCK2 O75116 1/20 0.36
KDM4E B2RXH2 1/20 0.35
MAPK1 P28482 1/20 0.35
HTT P42858 1/20 0.35
CYP3A4 P08684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL533862 0.86 REN (0.45) RENKCNH2KDM1ACHRNB2CHRNA4
SCHEMBL533861 0.86 REN (0.45) RENKCNH2KDM1ACHRNB2CHRNA4
SCHEMBL534503 0.76 REN (0.36) RENKCNH2CYP3A4
SCHEMBL534505 0.76 REN (0.36) RENKCNH2CYP3A4
SCHEMBL534504 0.76 REN (0.36) RENKCNH2CYP3A4
SCHEMBL534498 0.74 SPR (0.43) RENKCNH2MEN1KMT2AKDM4E
SCHEMBL7869553 0.73 REN (0.71) RENKCNH2KDM1ACYP2D6CYP3A4
SCHEMBL556570 0.72 SLC6A4 (0.32) RENKCNH2MEN1KMT2ASMN1; SMN2
SCHEMBL556569 0.72 SLC6A4 (0.32) RENKCNH2MEN1KMT2ASMN1; SMN2
SCHEMBL556568 0.72 SLC6A4 (0.32) RENKCNH2MEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2413941-A1 RENIN INHIBITORS Merck Sharp & Dohme Corp. (US) 2012-02-08 EP disclosed
WO-2010114978-A1 RENIN INHIBITORS MERCK SHARP & DOHME CORP. (US) 2010-10-07 WO disclosed