SCHEMBL533911

SCHEMBL533911

Cc1cc(-c2ccccc2CCNC(=O)OCc2ccccc2)ccc1C1CNCCC1=O

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
REN P00797 12/20 0.48
KCNH2 Q12809 11/20 0.48
L3MBTL1 Q9Y468 1/20 0.41
IDO1 P14902 2/20 0.41
CD274 Q9NZQ7 1/20 0.41
CYP3A4 P08684 1/20 0.40
ENPP2 Q13822 1/20 0.40
TRPM8 Q7Z2W7 1/20 0.39
PTGER4 P35408 1/20 0.38
PTGER3 P43115 1/20 0.38
GAA P10253 1/20 0.38
TDO2 P48775 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL534760 0.86 REN (0.60) RENKCNH2CYP3A4
SCHEMBL556192 0.80 ABCB1 (0.39) RENKCNH2L3MBTL1CD274ENPP2
SCHEMBL10202500 0.80 REN (0.56) RENKCNH2L3MBTL1CYP3A4ENPP2
SCHEMBL556382 0.76 REN (0.39) RENKCNH2L3MBTL1IDO1CD274
SCHEMBL7863795 0.73 REN (0.54) RENKCNH2CYP3A4
SCHEMBL533903 0.70 REN (0.46) RENKCNH2CD274CYP3A4
SCHEMBL7863764 0.69 REN (0.58) RENKCNH2CYP3A4
SCHEMBL10202506 0.68 REN (0.63) RENKCNH2CYP3A4
SCHEMBL7872527 0.68 REN (0.61) RENKCNH2CYP3A4
SCHEMBL7870969 0.67 REN (0.49) RENKCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2413941-A1 RENIN INHIBITORS Merck Sharp & Dohme Corp. (US) 2012-02-08 EP disclosed
WO-2010114978-A1 RENIN INHIBITORS MERCK SHARP & DOHME CORP. (US) 2010-10-07 WO disclosed