SCHEMBL534760

SCHEMBL534760

CC(=O)NCCc1ccccc1-c1ccc(C2CNCCC2=O)c(C)c1

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
REN P00797 18/20 0.60
KCNH2 Q12809 17/20 0.60
CYP3A4 P08684 6/20 0.52
MTNR1A P48039 1/20 0.41
MTNR1B P49286 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL533911 0.86 REN (0.48) RENKCNH2CYP3A4
SCHEMBL7863764 0.82 REN (0.58) RENKCNH2CYP3A4MTNR1AMTNR1B
SCHEMBL7872527 0.81 REN (0.61) RENKCNH2CYP3A4MTNR1AMTNR1B
SCHEMBL533903 0.80 REN (0.46) RENKCNH2CYP3A4MTNR1AMTNR1B
SCHEMBL10202485 0.77 REN (0.69) RENKCNH2CYP3A4
SCHEMBL10202479 0.77 REN (0.69) RENKCNH2CYP3A4
SCHEMBL557035 0.76 REN (0.43) RENKCNH2CYP3A4MTNR1AMTNR1B
SCHEMBL7873280 0.75 REN (0.85) RENKCNH2CYP3A4
SCHEMBL10202561 0.75 REN (1.00) RENKCNH2CYP3A4
SCHEMBL7871265 0.75 REN (0.85) RENKCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2413941-A1 RENIN INHIBITORS Merck Sharp & Dohme Corp. (US) 2012-02-08 EP disclosed
WO-2010114978-A1 RENIN INHIBITORS MERCK SHARP & DOHME CORP. (US) 2010-10-07 WO disclosed