SCHEMBL5339664

SCHEMBL5339664

O=C(O)c1c(-c2ccccc2)c2ccccc2n2ccnc12

nearest known ligand 0.59

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 7/20 0.59
AGTR1 P30556 3/20 0.46
PTGS2 P35354 1/20 0.43
KMT2A Q03164 2/20 0.43
PADI4 Q9UM07 1/20 0.42
LMNA P02545 2/20 0.41
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
CCNE1 P24864 1/20 0.39
CDK2 P24941 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
HPGD P15428 1/20 0.39
IDO1 P14902 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31636947 0.83 TACR1 (0.45) TACR1KMT2ALMNAKDM4EALDH1A1
SCHEMBL5342544 0.81 TACR1 (0.52) TACR1KMT2ALMNAKDM4EALDH1A1
SCHEMBL7324607 0.80 IDO1 (0.43) TACR1AGTR1PTGS2LMNAKDM4E
SCHEMBL14463630 0.78 PTGS2 (0.58) TACR1AGTR1PTGS2KMT2APADI4
SCHEMBL31636783 0.74 TACR1 (0.43) TACR1PDE3BPDE3ACCNE1CDK2
SCHEMBL5470895 0.73 TACR1 (1.00) TACR1
SCHEMBL5335958 0.73 TACR1 (0.58) TACR1AGTR1PTGS2KMT2APADI4
SCHEMBL4494163 0.72 TACR1 (0.59) TACR1AGTR1KMT2ALMNAKDM4E
SCHEMBL31636422 0.70 EGLN1 (0.55) TACR1KMT2ALMNAKDM4EALDH1A1
SCHEMBL29636632 0.70 MAPK8 (0.41) TACR1PDE3BPDE3ACCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007074491-A1 HETEROTRICYCLIC AMIDE DERIVATIVES AS NEUROKININ-l (NKl) RECEPTOR LIGANDS UNIVERSITA DEGLI STUDI DI SIENA (IT) 2007-07-05 WO disclosed
WO-2007074491-A1 HETEROTRICYCLIC AMIDE DERIVATIVES AS NEUROKININ-l (NKl) RECEPTOR LIGANDS UNIVERSITA DEGLI STUDI DI SIENA (IT) 2007-07-05 WO disclosed