SCHEMBL5335958

SCHEMBL5335958

O=C(O)c1c(-c2ccccc2)c2ccccc2n2cncc12

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 4/20 0.58
AGTR1 P30556 3/20 0.47
PTGS2 P35354 1/20 0.44
LMNA P02545 1/20 0.42
PADI4 Q9UM07 4/20 0.42
GABRA5 P31644 2/20 0.40
KMT2A Q03164 1/20 0.40
POLB P06746 2/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
BRD9 Q9H8M2 1/20 0.39
TDO2 P48775 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14463536 0.82 SMN1; SMN2 (0.54) TACR1LMNAKMT2AKDM4EALDH1A1
SCHEMBL14463630 0.79 PTGS2 (0.58) TACR1AGTR1PTGS2LMNAPADI4
SCHEMBL8597724 0.76 REN (0.41) TACR1LMNAKMT2AALDH1A1HPGD
SCHEMBL5339664 0.73 TACR1 (0.59) TACR1AGTR1PTGS2LMNAPADI4
SCHEMBL3356849 0.70 GABRA5 (0.50) GABRA5TDO2
SCHEMBL28322929 0.69 AGTR1 (0.50) AGTR1PTGS2LMNAPADI4KMT2A
SCHEMBL4494163 0.68 TACR1 (0.59) TACR1AGTR1LMNAKMT2APOLB
SCHEMBL2490336 0.65 AGTR1 (0.53) AGTR1LMNAKMT2APOLBKDM4E
SCHEMBL29262209 0.65 LMNA (0.55) AGTR1LMNAKMT2APOLBKDM4E
SCHEMBL10924110 0.64 GABRA5 (0.55) GABRA5KDM4EALDH1A1BRD9TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007074491-A1 HETEROTRICYCLIC AMIDE DERIVATIVES AS NEUROKININ-l (NKl) RECEPTOR LIGANDS UNIVERSITA DEGLI STUDI DI SIENA (IT) 2007-07-05 WO disclosed
WO-2007074491-A1 HETEROTRICYCLIC AMIDE DERIVATIVES AS NEUROKININ-l (NKl) RECEPTOR LIGANDS UNIVERSITA DEGLI STUDI DI SIENA (IT) 2007-07-05 WO disclosed