SCHEMBL534056

SCHEMBL534056

Cc1c(C2CCN(C(=O)O)CC2c2ccc(-c3ccccc3CCN)cc2Cl)cc[nH]c1=O

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
REN P00797 7/20 0.39
KCNH2 Q12809 6/20 0.39
CYP3A4 P08684 1/20 0.39
DPP4 P27487 3/20 0.32
DPP7 Q9UHL4 1/20 0.32
GHSR Q92847 1/20 0.31
KDM5B Q9UGL1 1/20 0.31
BRD9 Q9H8M2 3/20 0.31
KDM5A P29375 1/20 0.31
CHRM3 P20309 2/20 0.31
CHRM2 P08172 1/20 0.31
CHRM4 P08173 1/20 0.31
CHRM5 P08912 1/20 0.31
CHRM1 P11229 1/20 0.31
CD274 Q9NZQ7 1/20 0.30
PTGER1 P34995 1/20 0.30
PTGER4 P35408 1/20 0.30
PTGER3 P43115 1/20 0.30
PTGER2 P43116 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL534448 0.85 REN (0.48) RENKCNH2CYP3A4CD274PTGER1
SCHEMBL533938 0.84 REN (0.42) RENKCNH2CYP3A4DPP4DPP7
SCHEMBL534057 0.80 REN (0.58) RENKCNH2CYP3A4DPP4DPP7
SCHEMBL533961 0.79 SMN1; SMN2 (0.35) DPP4
SCHEMBL533953 0.78 REN (0.48) RENKCNH2CYP3A4DPP4CHRM3
SCHEMBL556088 0.72 REN (0.41) RENKCNH2CYP3A4DPP4DPP7
SCHEMBL534353 0.72 REN (0.37) RENKCNH2CYP3A4PTGER1PTGER4
SCHEMBL535442 0.70 REN (0.41) RENKCNH2CYP3A4CHRM3PTGER1
SCHEMBL535144 0.70 REN (0.74) RENKCNH2CYP3A4
SCHEMBL535443 0.70 REN (0.41) RENKCNH2CYP3A4CHRM3PTGER1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2413941-A1 RENIN INHIBITORS Merck Sharp & Dohme Corp. (US) 2012-02-08 EP disclosed
WO-2010114978-A1 RENIN INHIBITORS MERCK SHARP & DOHME CORP. (US) 2010-10-07 WO disclosed