SCHEMBL5344200

SCHEMBL5344200

CCOC(=O)c1[nH]ccc1NCc1nc2c(C)c(C)ccc2[nH]1.Cc1ccc2[nH]c(Cn3c(=S)[nH]c(=O)c4[nH]ccc43)nc2c1C

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MPO P05164 19/20 0.38
TPO P07202 18/20 0.38
KCNH2 Q12809 2/20 0.37
OPRM1 P35372 1/20 0.35
CYP3A4 P08684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1536713 0.84 ALDH1A1 (0.42) OPRM1
SCHEMBL1536751 0.83 MPO (0.47) MPOTPOKCNH2OPRM1CYP3A4
SCHEMBL1536842 0.68 MAPT (0.65)
SCHEMBL1536633 0.68 ALDH1A1 (0.48)
SCHEMBL1536749 0.64 MPO (0.61) MPOTPOKCNH2OPRM1CYP3A4
SCHEMBL1536767 0.63 NUDT1 (0.45)
SCHEMBL1536763 0.60 ALDH1A1 (0.39)
SCHEMBL1536617 0.60 MAPK8 (0.41)
SCHEMBL1536665 0.59 MPO (0.55) MPOTPOKCNH2OPRM1CYP3A4
SCHEMBL18557963 0.59 KMT2A (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1824855-A1 NOVEL PYRROLO [3, 2-D]PYRIMIDIN-4-ONE DERIVATIVES AND THEIR USE IN THERAPY AstraZeneca AB (SE) 2007-08-29 EP disclosed
WO-2006062465-A1 NOVEL PYRROLO [3, 2-D] PYRIMIDIN-4-ONE DERIVATIVES AND THEIR USE IN THERAPY ASTRAZENECA AB (SE) 2006-06-15 WO disclosed