SCHEMBL5344366

SCHEMBL5344366

Cc1ccc(-c2c(-c3ccc(F)cc3)nc3ncc(-c4cccc(C(F)(F)F)c4)cn23)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.43
NR3C1 P04150 1/20 0.43
PGR P06401 1/20 0.43
AKT1 P31749 3/20 0.43
AKT2 P31751 3/20 0.43
MAOB P27338 1/20 0.38
GRIN1 Q05586 2/20 0.38
GRIN2B Q13224 2/20 0.38
GSK3B P49841 1/20 0.37
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37
NPC1 O15118 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
MAPT P10636 1/20 0.37
CYP2C19 P33261 1/20 0.37
RAB9A P51151 1/20 0.37
KCNH2 Q12809 1/20 0.37
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5343214 0.95 TDP1 (0.47) TDP1NR3C1PGRAKT1AKT2
SCHEMBL5324596 0.93 TDP1 (0.46) TDP1NR3C1PGRAKT1AKT2
SCHEMBL5350061 0.90 TDP1 (0.39) TDP1NR3C1PGRAKT1AKT2
SCHEMBL5344952 0.90 TDP1 (0.45) TDP1NR3C1PGRAKT1AKT2
SCHEMBL5344560 0.89 MAPK14 (0.42) TDP1NR3C1PGRAKT1AKT2
SCHEMBL5354199 0.89 NR1H4 (0.44) TDP1NR3C1PGRAKT1AKT2
SCHEMBL5338540 0.85 AKT1 (0.46) TDP1NR3C1PGRAKT1AKT2
Hydrochloric Acid SCHEMBL5344599 0.84 AKT1 (0.45) TDP1NR3C1PGRAKT1AKT2
SCHEMBL5342580 0.83 TDP1 (0.47) TDP1NR3C1PGRMAOBGRIN1
SCHEMBL5354165 0.82 AKT1 (0.44) TDP1AKT1AKT2GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007096764-A2 BICYCLIC HETEROARYL DERIVATIVES AS CANNABINOID RECEPTOR MODULATORS GLENMARK PHARMACEUTICALS S.A. (US) 2007-08-30 WO claimed
WO-2007096764-A2 BICYCLIC HETEROARYL DERIVATIVES AS CANNABINOID RECEPTOR MODULATORS GLENMARK PHARMACEUTICALS S.A. (US) 2007-08-30 WO disclosed