SCHEMBL5344560

SCHEMBL5344560

CSc1ccc(-c2c(-c3ccc(F)cc3)nc3ncc(-c4cccc(C(F)(F)F)c4)cn23)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 5/20 0.42
MAPK13 O15264 4/20 0.42
MAPK12 P53778 4/20 0.42
MAPK11 Q15759 4/20 0.42
GCGR P47871 2/20 0.42
TDP1 Q9NUW8 2/20 0.41
NR3C1 P04150 1/20 0.41
PGR P06401 1/20 0.41
AKT1 P31749 2/20 0.41
AKT2 P31751 2/20 0.41
PTGS1 P23219 2/20 0.41
PTGS2 P35354 2/20 0.41
ALDH1A1 P00352 2/20 0.37
GAA P10253 1/20 0.37
ATM Q13315 1/20 0.37
LMNA P02545 1/20 0.37
DYRK3 O43781 1/20 0.37
CCNT1 O60563 1/20 0.37
CCNA2 P20248 1/20 0.37
CDK2 P24941 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5343214 0.92 TDP1 (0.47) MAPK14MAPK13MAPK12MAPK11TDP1
SCHEMBL5319387 0.91 AKT1 (0.41) MAPK14TDP1AKT1AKT2PTGS1
SCHEMBL5324596 0.90 TDP1 (0.46) MAPK14MAPK13MAPK12MAPK11TDP1
SCHEMBL5344366 0.89 TDP1 (0.43) TDP1NR3C1PGRAKT1AKT2
SCHEMBL5344952 0.87 TDP1 (0.45) TDP1NR3C1PGRAKT1AKT2
SCHEMBL5354199 0.86 NR1H4 (0.44) TDP1NR3C1PGRAKT1AKT2
SCHEMBL5338540 0.83 AKT1 (0.46) TDP1NR3C1PGRAKT1AKT2
Hydrochloric Acid SCHEMBL5344599 0.82 AKT1 (0.45) TDP1NR3C1PGRAKT1AKT2
SCHEMBL5320666 0.81 MAPK14 (0.43) MAPK14MAPK13MAPK12MAPK11GCGR
SCHEMBL5342580 0.81 TDP1 (0.47) TDP1NR3C1PGRALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007096764-A2 BICYCLIC HETEROARYL DERIVATIVES AS CANNABINOID RECEPTOR MODULATORS GLENMARK PHARMACEUTICALS S.A. (US) 2007-08-30 WO claimed
WO-2007096764-A2 BICYCLIC HETEROARYL DERIVATIVES AS CANNABINOID RECEPTOR MODULATORS GLENMARK PHARMACEUTICALS S.A. (US) 2007-08-30 WO disclosed