SCHEMBL5344952

SCHEMBL5344952

Fc1ccc(-c2nc3ncc(-c4cccc(C(F)(F)F)c4)cn3c2-c2cc(F)cc(F)c2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.45
NR3C1 P04150 1/20 0.45
PGR P06401 1/20 0.45
AKT1 P31749 1/20 0.42
AKT2 P31751 1/20 0.42
MAOB P27338 1/20 0.39
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
GRIN1 Q05586 5/20 0.37
GRIN2B Q13224 5/20 0.37
PARP1 P09874 1/20 0.36
TRPA1 O75762 1/20 0.36
ALDH1A1 P00352 2/20 0.35
GAA P10253 2/20 0.35
KDM4E B2RXH2 2/20 0.35
ATM Q13315 1/20 0.35
DYRK1A Q13627 1/20 0.35
DYRK2 Q92630 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5343214 0.95 TDP1 (0.47) TDP1NR3C1PGRAKT1AKT2
SCHEMBL5324596 0.93 TDP1 (0.46) TDP1NR3C1PGRAKT1AKT2
SCHEMBL5344366 0.90 TDP1 (0.43) TDP1NR3C1PGRAKT1AKT2
SCHEMBL5354199 0.87 NR1H4 (0.44) TDP1NR3C1PGRAKT1AKT2
SCHEMBL5344560 0.87 MAPK14 (0.42) TDP1NR3C1PGRAKT1AKT2
SCHEMBL5338540 0.85 AKT1 (0.46) TDP1NR3C1PGRAKT1AKT2
SCHEMBL5342580 0.85 TDP1 (0.47) TDP1NR3C1PGRMAOBADORA2A
Hydrochloric Acid SCHEMBL5344599 0.84 AKT1 (0.45) TDP1NR3C1PGRAKT1AKT2
SCHEMBL5346776 0.81 AKT1 (0.42) TDP1AKT1AKT2MAOBADORA2A
SCHEMBL5350061 0.80 TDP1 (0.39) TDP1NR3C1PGRAKT1AKT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007096764-A2 BICYCLIC HETEROARYL DERIVATIVES AS CANNABINOID RECEPTOR MODULATORS GLENMARK PHARMACEUTICALS S.A. (US) 2007-08-30 WO disclosed