SCHEMBL5344648

SCHEMBL5344648

CCC(C)C1=NN(C(C)C)C(=O)N(c2ccc(CC3=NCCN3)cc2)c2cc(C)c(OCc3ccccc3)cc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTH1R Q03431 4/20 0.51
NISCH Q9Y2I1 6/20 0.39
HTR1D P28221 3/20 0.38
HTR1B P28222 2/20 0.38
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
ADRA1D P25100 3/20 0.36
ADRA1A P35348 3/20 0.36
ADRA1B P35368 3/20 0.36
TAAR1 Q96RJ0 2/20 0.36
LMNA P02545 1/20 0.36
CYP1A2 P05177 1/20 0.36
ADRA2A P08913 1/20 0.36
CYP2D6 P10635 1/20 0.36
TSHR P16473 1/20 0.36
ADRA2B P18089 1/20 0.36
ADRA2C P18825 1/20 0.36
CYP3A4 P08684 1/20 0.34
KCNH2 Q12809 1/20 0.34
MCHR1 Q99705 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5324368 0.86 PTH1R (0.67) PTH1RNISCHHTR1DHTR1BMAOA
SCHEMBL5350284 0.84 PTH1R (0.39) PTH1RMAOAMAOB
SCHEMBL5376690 0.75 PTH1R (0.74) PTH1RCYP3A4KCNH2MCHR1
SCHEMBL5487298 0.74 PTH1R (0.67) PTH1RHTR1DHTR1B
SCHEMBL5358731 0.74 PTH1R (0.53) PTH1RNISCHHTR1DHTR1BMAOA
SCHEMBL5368169 0.72 PTH1R (0.69) PTH1RADRA1DADRA1AADRA1BTAAR1
SCHEMBL5352432 0.72 PTH1R (0.33) PTH1RMAOB
SCHEMBL5363635 0.70 PTH1R (0.82) PTH1RHTR1DHTR1B
SCHEMBL5367699 0.70 PTH1R (0.76) PTH1RHTR1DHTR1B
SCHEMBL5362367 0.70 PTH1R (0.84) PTH1RHTR1DHTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007135417-A1 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2007-11-29 WO disclosed