SCHEMBL5346572

SCHEMBL5346572

CC(C)COc1cccc2onc(OCC3CCN(CCC4(C(=O)O)CCOC(C)C4)CC3)c12

nearest known ligand 0.62

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 15/20 0.62
CYP3A4 P08684 1/20 0.46
ACHE P22303 1/20 0.37
KCNH2 Q12809 3/20 0.32
HTR2A P28223 2/20 0.32
HTR1D P28221 2/20 0.32
HTR7 P34969 1/20 0.32
HTR2B P41595 1/20 0.32
HTR1A P08908 1/20 0.31
HTR1B P28222 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5341243 0.92 HTR4 (0.60) HTR4CYP3A4ACHEKCNH2HTR2A
SCHEMBL5112331 0.90 HTR4 (0.72) HTR4CYP3A4ACHEKCNH2HTR2A
SCHEMBL5349482 0.89 HTR4 (0.53) HTR4CYP3A4ACHEKCNH2
SCHEMBL5116914 0.85 HTR4 (0.70) HTR4CYP3A4ACHEKCNH2HTR2A
SCHEMBL5394346 0.84 HTR4 (0.55) HTR4CYP3A4ACHE
SCHEMBL5112304 0.84 HTR4 (0.79) HTR4CYP3A4ACHEKCNH2
SCHEMBL5112375 0.83 HTR4 (0.71) HTR4CYP3A4ACHEKCNH2
SCHEMBL5122071 0.83 HTR4 (0.71) HTR4CYP3A4ACHEKCNH2
SCHEMBL15949468 0.82 HTR4 (0.74) HTR4CYP3A4ACHEKCNH2HTR2A
SCHEMBL5334028 0.82 HTR4 (0.57) HTR4CYP3A4ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1856114-A1 BENZISOXAZOLE DERIVATIVES Pfizer, Inc. (US) 2007-11-21 EP disclosed
WO-2006090224-A1 BENZISOXAZOLE DERIVATIVES PFIZER JAPAN INC. (JP) 2006-08-31 WO disclosed