SCHEMBL5349482

SCHEMBL5349482

CC1CC(CCN2CCC(COc3noc4cccc(OCC(F)(F)F)c34)CC2)(C(=O)O)CCO1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 11/20 0.53
CYP3A4 P08684 1/20 0.46
ACHE P22303 1/20 0.36
DRD3 P35462 1/20 0.34
DCPS Q96C86 1/20 0.33
DRD2 P14416 1/20 0.32
DRD4 P21917 1/20 0.32
HCRTR2 O43614 1/20 0.32
KCNH2 Q12809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5334028 0.93 HTR4 (0.57) HTR4CYP3A4ACHEDCPSHCRTR2
SCHEMBL5341243 0.91 HTR4 (0.60) HTR4CYP3A4ACHEKCNH2
SCHEMBL5120856 0.90 HTR4 (0.60) HTR4CYP3A4ACHEDRD3DCPS
SCHEMBL5346572 0.89 HTR4 (0.62) HTR4CYP3A4ACHEKCNH2
SCHEMBL5119519 0.85 HTR4 (0.60) HTR4CYP3A4ACHEDRD3DCPS
SCHEMBL5394346 0.84 HTR4 (0.55) HTR4CYP3A4ACHE
SCHEMBL5114319 0.84 HTR4 (0.66) HTR4CYP3A4ACHEDCPSHCRTR2
SCHEMBL5348518 0.84 HTR4 (0.53) HTR4CYP3A4ACHEDRD3KCNH2
Hydrochloric Acid SCHEMBL17275530 0.83 HTR4 (0.65) HTR4CYP3A4ACHEDCPSHCRTR2
SCHEMBL17275529 0.83 HTR4 (0.65) HTR4CYP3A4ACHEDCPSHCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1856114-A1 BENZISOXAZOLE DERIVATIVES Pfizer, Inc. (US) 2007-11-21 EP disclosed
WO-2006090224-A1 BENZISOXAZOLE DERIVATIVES PFIZER JAPAN INC. (JP) 2006-08-31 WO disclosed