SCHEMBL534711

SCHEMBL534711

NC(=O)CCCc1ccccc1C#CBr

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 10/20 0.40
MTNR1A P48039 1/20 0.40
MPO P05164 3/20 0.38
FFAR4 Q5NUL3 3/20 0.37
TLR8 Q9NR97 1/20 0.36
ATM Q13315 1/20 0.36
SLC6A4 P31645 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TSPO P30536 1/20 0.35
DRD3 P35462 1/20 0.35
HDAC3 O15379 1/20 0.34
MAPK1 P28482 1/20 0.34
ADRA1A P35348 1/20 0.34
HDAC4 P56524 1/20 0.34
SLC6A3 Q01959 1/20 0.34
HDAC1 Q13547 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC10 Q969S8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29045424 0.81 FFAR1 (0.46) FFAR1MTNR1AMPOFFAR4TLR8
SCHEMBL30828055 0.75 TAAR1 (0.53) FFAR1MTNR1AMPOFFAR4TLR8
SCHEMBL6800944 0.74 MTNR1A (0.40) FFAR1MTNR1AMPOFFAR4MAPK1
SCHEMBL27530341 0.73 TAAR1 (0.55) MTNR1AMPOSLC6A4ALDH1A1
SCHEMBL3790529 0.73 FDPS (0.44) MTNR1AMPOTLR8ATMSLC6A4
SCHEMBL517084 0.72 CYP4F2 (0.49) MTNR1AMPOTLR8HDAC1HDAC2
SCHEMBL5878486 0.72 CYP4F2 (0.49) MTNR1AMPOTLR8HDAC1HDAC2
SCHEMBL29407477 0.72 CYP4F2 (0.49) MTNR1AMPOTLR8HDAC1HDAC2
SCHEMBL9395052 0.72 CYP4F2 (0.49) MTNR1AMPOTLR8HDAC1HDAC2
Hydrochloric Acid SCHEMBL10784054 0.72 FDPS (0.43) MTNR1AMPOTLR8ATMSLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2413941-A1 RENIN INHIBITORS Merck Sharp & Dohme Corp. (US) 2012-02-08 EP disclosed
WO-2010114978-A1 RENIN INHIBITORS MERCK SHARP & DOHME CORP. (US) 2010-10-07 WO disclosed