SCHEMBL5347690

SCHEMBL5347690

COc1cccc(C(C)N2CCN(c3c(C)c(C)c4c(c3C)C(N3CCCC3)C(C)(C)O4)CC2)c1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.36
ACHE P22303 5/20 0.36
MBTD1 Q05BQ5 1/20 0.35
L3MBTL3 Q96JM7 1/20 0.35
ALDH1A1 P00352 1/20 0.35
IDH1 O75874 1/20 0.33
OGA O60502 3/20 0.32
POLB P06746 1/20 0.32
ROCK2 O75116 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM1 P11229 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5346017 0.99 HSD11B1 (0.36) HSD11B1ACHEMBTD1L3MBTL3ALDH1A1
SCHEMBL5343241 0.89 CHRM2 (0.41) HSD11B1ACHEALDH1A1OGACHRM2
Hydrochloric Acid SCHEMBL5343678 0.88 CHRM2 (0.41) HSD11B1ACHEALDH1A1OGACHRM2
SCHEMBL5350819 0.86 TSHR (0.41) ALDH1A1POLBMEN1KMT2A
Hydrochloric Acid SCHEMBL5339938 0.86 CYP2D6 (0.40) MBTD1L3MBTL3ALDH1A1CHRM2CHRM1
SCHEMBL5347702 0.80 HSD11B1 (0.35) HSD11B1ACHE
SCHEMBL5347696 0.80 HRH3 (0.51)
Hydrochloric Acid SCHEMBL5346025 0.80 HSD11B1 (0.35) HSD11B1ACHE
Hydrochloric Acid SCHEMBL5346020 0.79 HRH3 (0.50)
SCHEMBL5344095 0.79 ALDH1A1 (0.40) ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7208495-B2 Benzo-fused 5-membered hetrocycle compounds, process for preparation of the same, and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-04-24 US claimed