SCHEMBL5347702

SCHEMBL5347702

COc1cccc(C(C)N2CCN(c3c(C)c(C)c4c(c3C)C(C3CCNC3)C(C)(C)O4)CC2)c1

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.35
PIM1 P11309 1/20 0.32
ACHE P22303 3/20 0.31
CFTR P13569 1/20 0.31
AURKA O14965 1/20 0.30
SLC6A2 P23975 3/20 0.30
SLC6A4 P31645 2/20 0.30
SLC6A3 Q01959 1/20 0.30
ADRB1 P08588 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5346025 0.99 HSD11B1 (0.35) HSD11B1PIM1ACHECFTRAURKA
SCHEMBL5343256 0.91 CHRM2 (0.35) HSD11B1
Hydrochloric Acid SCHEMBL5343688 0.90 CHRM2 (0.35) HSD11B1
SCHEMBL5347690 0.80 HSD11B1 (0.36) HSD11B1ACHE
Hydrochloric Acid SCHEMBL5346017 0.79 HSD11B1 (0.36) HSD11B1ACHE
SCHEMBL5343241 0.71 CHRM2 (0.41) HSD11B1ACHE
Hydrochloric Acid SCHEMBL5344037 0.70 MAPT (0.34)
SCHEMBL2472859 0.68 SLC18A3 (0.41) ADRB1
SCHEMBL5350943 0.68 KCNH2 (0.44) ADRB1
Hydrochloric Acid SCHEMBL5339938 0.68 CYP2D6 (0.40) AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7208495-B2 Benzo-fused 5-membered hetrocycle compounds, process for preparation of the same, and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-04-24 US claimed