SCHEMBL5343256

SCHEMBL5343256

COc1ccc(C(C)N2CCN(c3c(C)c(C)c4c(c3C)C(C3CCNC3)C(C)(C)O4)CC2)cc1

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 4/20 0.35
CHRM1 P11229 2/20 0.35
CHRM4 P08173 1/20 0.35
CHRM3 P20309 1/20 0.35
OPRM1 P35372 2/20 0.33
HSD11B1 P28845 3/20 0.33
OGA O60502 1/20 0.31
USP2 O75604 1/20 0.30
LMNA P02545 1/20 0.30
TSHR P16473 1/20 0.30
HTT P42858 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5343688 0.99 CHRM2 (0.35) CHRM2CHRM1CHRM4CHRM3OPRM1
SCHEMBL5347702 0.91 HSD11B1 (0.35) HSD11B1
Hydrochloric Acid SCHEMBL5346025 0.90 HSD11B1 (0.35) HSD11B1
Hydrochloric Acid SCHEMBL5339945 0.89 CYP2D6 (0.36) CHRM2CHRM1OPRM1ALDH1A1
SCHEMBL5343241 0.79 CHRM2 (0.41) CHRM2CHRM1CHRM4CHRM3OPRM1
Hydrochloric Acid SCHEMBL5343678 0.79 CHRM2 (0.41) CHRM2CHRM1CHRM4CHRM3OPRM1
SCHEMBL2472859 0.75 SLC18A3 (0.41) LMNATSHRHTTALDH1A1KMT2A
Hydrochloric Acid SCHEMBL5344037 0.73 MAPT (0.34) KDM4E
SCHEMBL5351949 0.72 LMNA (0.35) LMNAALDH1A1
SCHEMBL5347690 0.70 HSD11B1 (0.36) CHRM2CHRM1HSD11B1OGAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7208495-B2 Benzo-fused 5-membered hetrocycle compounds, process for preparation of the same, and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-04-24 US claimed