SCHEMBL5354411

SCHEMBL5354411

CS(=O)(=O)Nc1ccc(C(=O)CCC(=O)O)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.56
PTGS2 P35354 4/20 0.54
HPGD P15428 2/20 0.54
RECQL P46063 1/20 0.54
HDAC3 O15379 1/20 0.52
HDAC4 P56524 1/20 0.52
HDAC1 Q13547 1/20 0.52
HDAC7 Q8WUI4 1/20 0.52
HDAC2 Q92769 1/20 0.52
HDAC10 Q969S8 1/20 0.52
HDAC11 Q96DB2 1/20 0.52
HDAC8 Q9BY41 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
HDAC9 Q9UKV0 1/20 0.52
HDAC5 Q9UQL6 1/20 0.52
NR4A2 P43354 1/20 0.52
USP5 P45974 1/20 0.51
LMNA P02545 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
L3MBTL1 Q9Y468 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9447463 0.90 PDE4B (0.54) KMT2APTGS2HPGDRECQLHDAC3
SCHEMBL7243169 0.85 HPGD (0.53) KMT2APTGS2HPGDRECQLHDAC3
SCHEMBL5352346 0.84 HPGD (0.55) KMT2APTGS2HPGDRECQLHDAC3
SCHEMBL9447401 0.83 HPGD (0.54) KMT2APTGS2HPGDRECQLHDAC3
SCHEMBL9078412 0.83 HPGD (0.54) KMT2APTGS2HPGDRECQLHDAC3
SCHEMBL8203459 0.81 HPGD (0.52) KMT2APTGS2HPGDRECQLHDAC3
SCHEMBL1474479 0.81 HPGD (0.63) KMT2APTGS2HPGDRECQLHDAC3
SCHEMBL11818687 0.81 THRA (0.65) KMT2AHPGDRECQLHDAC3HDAC4
SCHEMBL9657514 0.81 HPGD (0.51) KMT2APTGS2HPGDRECQLHDAC3
Hydrochloric Acid SCHEMBL11815733 0.80 GSR (0.66) KMT2AHPGDRECQLHDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1328253-C Fumaric acid ibutilide synthesis method ZHEJIANG JIUXU PHARMACEUTICAL (CN) 2007-07-25 CN disclosed
US-7232930-B2 Compounds and methods for preparing methanesulfonamides PHARMACIA & UPJOHN COMPANY (US) 2007-06-19 US disclosed
US-7232930-B2 Compounds and methods for preparing methanesulfonamides PHARMACIA & UPJOHN COMPANY (US) 2007-06-19 US disclosed
US-7232930-B2 Compounds and methods for preparing methanesulfonamides PHARMACIA & UPJOHN COMPANY (US) 2007-06-19 US disclosed
CN-1733714-A Fumaric acid ibutilide synthesis method ZHEJIANG JIUXU PHARMACEUTICAL (CN) 2006-02-15 CN disclosed
EP-1395549-A1 COMPOUNDS AND METHODS FOR PREPARING METHANESULFONAMIDES PHARMACIA & UPJOHN COMPANY (US) 2004-03-10 EP disclosed
WO-2002098845-A1 COMPOUNDS AND METHODS FOR PREPARING METHANESULFONAMIDES PHARMACIA & UPJOHN COMPANY (US) 2002-12-12 WO disclosed
EP-0802900-B1 ANTIARRHYTHMIC (S)-ENANTIOMERS OF METHANESULFONAMIDES UPJOHN CO (US) 2000-02-16 EP disclosed
US-5874475-A DO NOT HAVE SIDE EFFECT OF PRODUCING POLYMORPHIC VENTRICULAR TACHYCARDIA PHARMACIA & UPJOHN COMPANY (US) 1999-02-23 US disclosed
EP-0802900-A1 ANTIARRHYTHMIC (S)-ENANTIOMERS OF METHANESULFONAMIDES PHARMACIA & UPJOHN COMPANY (US) 1997-10-29 EP disclosed
WO-1996021643-A1 ANTIARRHYTHMIC (S)-ENANTIOMERS OF METHANESULFONAMIDES PHARMACIA & UPJOHN COMPANY (US) 1996-07-18 WO disclosed
US-5405997-A Stable against rapid metabolism THE UPJOHN COMPANY (US) 1995-04-11 US disclosed
EP-0484378-B1 ANTIARRHYTHMIC TERTIARY AMINE-ALKENYL-PHENYL-ALKANESULFONAMIDES UPJOHN CO (US) 1994-09-14 EP disclosed
US-5246946-A Antiarrhythmia agents and cardiovascular disorders EISAI CO., LTD. (JP) 1993-09-21 US disclosed
EP-0304888-B1 SULFONAMIDOLPHENYL DERIVATES AND THERAPEUTIC AND PREVENTIVE AGENTS FOR ARRYTHMIA CONTAINING SAME Eisai Co., Ltd. (JP) 1992-11-11 EP disclosed
US-5162347-A Piperidine derivatives and therapeutic and preventive agents for arrhythmia containing same EISAI CO., LTD. (JP) 1992-11-10 US disclosed
US-5155268-A Antiarrhythmic N-aminoalkylene alkyl and aryl sulfonamides THE UPJOHN COMPANY (US) 1992-10-13 US disclosed
US-5082850-A PIPERIDINE DERIVATIVES AND THERAPEUTIC AND PREVENTIVE AGENTS FOR ARRHYTHMIA CONTAINING SAME EISAI CO., LTD. (JP) 1992-01-21 US disclosed
US-4977165-A Piperidine derivative and therapeutic and preventive agents for arrhythmia containing same EISAI CO., LTD. (JP) 1990-12-11 US disclosed
EP-0304888-A1 Sulfonamidolphenyl derivates and therapeutic and preventive agents for arrythmia containing same Eisai Co., Ltd. (JP) 1989-03-01 EP disclosed