SCHEMBL8203459

SCHEMBL8203459

CCNC(=O)CCC(=O)c1ccc(NS(C)(=O)=O)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.52
RECQL P46063 1/20 0.52
HDAC3 O15379 1/20 0.51
HDAC4 P56524 1/20 0.51
HDAC1 Q13547 1/20 0.51
HDAC7 Q8WUI4 1/20 0.51
HDAC2 Q92769 1/20 0.51
HDAC10 Q969S8 1/20 0.51
HDAC11 Q96DB2 1/20 0.51
HDAC8 Q9BY41 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51
HDAC9 Q9UKV0 1/20 0.51
HDAC5 Q9UQL6 1/20 0.51
MEN1 O00255 4/20 0.49
KMT2A Q03164 4/20 0.49
PTGS2 P35354 3/20 0.46
CYP2C9 P11712 1/20 0.45
KDM4E B2RXH2 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
EPHX2 P34913 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5354411 0.81 KMT2A (0.56) HPGDRECQLHDAC3HDAC4HDAC1
SCHEMBL9447401 0.81 HPGD (0.54) HPGDRECQLHDAC3HDAC4HDAC1
SCHEMBL7243169 0.80 HPGD (0.53) HPGDRECQLHDAC3HDAC4HDAC1
SCHEMBL11949250 0.80 SMN1; SMN2 (0.61) HPGDRECQLMEN1KMT2AKDM4E
SCHEMBL1474479 0.79 HPGD (0.63) HPGDRECQLHDAC3HDAC4HDAC1
SCHEMBL5352346 0.79 HPGD (0.55) HPGDRECQLHDAC3HDAC4HDAC1
SCHEMBL9078412 0.78 HPGD (0.54) HPGDRECQLHDAC3HDAC4HDAC1
SCHEMBL8763454 0.78 GRIN1 (0.65) HPGDHDAC1HDAC8KDM4ESMN1; SMN2
SCHEMBL8203484 0.76 LMNA (0.53) HPGDRECQLMEN1KMT2ACYP2C9
SCHEMBL11818687 0.76 THRA (0.65) HPGDRECQLHDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0802900-B1 ANTIARRHYTHMIC (S)-ENANTIOMERS OF METHANESULFONAMIDES UPJOHN CO (US) 2000-02-16 EP disclosed
US-5874475-A DO NOT HAVE SIDE EFFECT OF PRODUCING POLYMORPHIC VENTRICULAR TACHYCARDIA PHARMACIA & UPJOHN COMPANY (US) 1999-02-23 US disclosed
EP-0802900-A1 ANTIARRHYTHMIC (S)-ENANTIOMERS OF METHANESULFONAMIDES PHARMACIA & UPJOHN COMPANY (US) 1997-10-29 EP disclosed
WO-1996021643-A1 ANTIARRHYTHMIC (S)-ENANTIOMERS OF METHANESULFONAMIDES PHARMACIA & UPJOHN COMPANY (US) 1996-07-18 WO disclosed
US-5405997-A Stable against rapid metabolism THE UPJOHN COMPANY (US) 1995-04-11 US disclosed
EP-0484378-B1 ANTIARRHYTHMIC TERTIARY AMINE-ALKENYL-PHENYL-ALKANESULFONAMIDES UPJOHN CO (US) 1994-09-14 EP disclosed
EP-0484378-A1 ANTIARRHYTHMIC TERTIARY AMINE-ALKENYL-PHENYL-ALKANESULFONAMIDES. UPJOHN CO (US) 1992-05-13 EP disclosed
WO-1991001299-A1 ANTIARRHYTHMIC TERTIARY AMINE-ALKENYL-PHENYL-ALKANESULFONAMIDES THE UPJOHN COMPANY (US) 1991-02-07 WO disclosed