SCHEMBL5355458

SCHEMBL5355458

NC1CCN(S(=O)(=O)c2ccc3[nH]c(-c4cc5c(F)cccc5[nH]c4=O)cc3c2Cl)C1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDR P35968 6/20 0.54
ALOX5AP P20292 5/20 0.39
FEN1 P39748 5/20 0.39
CHEK1 O14757 2/20 0.38
TDP1 Q9NUW8 1/20 0.35
DAO P14920 1/20 0.35
DDO Q99489 1/20 0.35
TRPV4 Q9HBA0 1/20 0.35
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
PDK1 Q15118 1/20 0.33
PDK2 Q15119 1/20 0.33
PDK3 Q15120 1/20 0.33
PDK4 Q16654 1/20 0.33
SSTR2 P30874 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5362169 0.84 KDR (0.77) KDRALOX5APFEN1CHEK1TDP1
SCHEMBL5355082 0.78 KDR (0.73) KDRALOX5APFEN1CHEK1
SCHEMBL5355698 0.70 KDR (1.00) KDRCHEK1
SCHEMBL5358982 0.69 KDR (0.89) KDRCHEK1
SCHEMBL5362580 0.67 KDR (0.70) KDRALOX5APFEN1CHEK1TDP1
SCHEMBL5359215 0.64 KDR (0.67) KDRALOX5APFEN1CHEK1TDP1
SCHEMBL15942385 0.62 DAO (0.53) KDRCHEK1DAODDO
SCHEMBL5355363 0.62 KDR (0.85) KDRCHEK1
SCHEMBL5367711 0.60 KDR (0.70) KDRCHEK1
SCHEMBL6795564 0.60 MEN1 (0.60) CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7169788-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2007-01-30 US disclosed
US-7169788-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2007-01-30 US disclosed
US-7169788-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2007-01-30 US disclosed