Predicted protein targets (top 20)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | TSHR | P16473 | 2/20 | 0.49 |
| ▸ | APOBEC3A | P31941 | 1/20 | 0.49 |
| ▸ | HTT | P42858 | 1/20 | 0.49 |
| ▸ | APOBEC3G | Q9HC16 | 1/20 | 0.49 |
| ▸ | MAPK1 | P28482 | 1/20 | 0.46 |
| ▸ | ALOX15 | P16050 | 1/20 | 0.46 |
| ▸ | SIRT2 | Q8IXJ6 | 1/20 | 0.46 |
| ▸ | SIRT1 | Q96EB6 | 1/20 | 0.46 |
| ▸ | SIRT3 | Q9NTG7 | 1/20 | 0.46 |
| ▸ | PARP1 | P09874 | 1/20 | 0.45 |
| ▸ | CYP1A2 | P05177 | 1/20 | 0.44 |
| ▸ | CYP3A4 | P08684 | 1/20 | 0.44 |
| ▸ | CYP2C9 | P11712 | 1/20 | 0.44 |
| ▸ | CYP2C19 | P33261 | 1/20 | 0.44 |
| ▸ | ALDH1A1 | P00352 | 3/20 | 0.44 |
| ▸ | KMT2A | Q03164 | 1/20 | 0.44 |
| ▸ | PARP15 | Q460N3 | 1/20 | 0.44 |
| ▸ | PARP10 | Q53GL7 | 1/20 | 0.44 |
| ▸ | HPGD | P15428 | 2/20 | 0.44 |
| ▸ | KDM4E | B2RXH2 | 1/20 | 0.44 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL31281188 | 1.00 | TSHR (0.49) | TSHRAPOBEC3AHTTAPOBEC3GMAPK1 | |
| Hydrochloric Acid SCHEMBL22445134 | 0.98 | TSHR (0.47) | TSHRAPOBEC3AHTTAPOBEC3GMAPK1 | |
| SCHEMBL18288064 | 0.85 | ALOX15 (0.55) | TSHRHTTALOX15CYP1A2CYP2C19 | |
| SCHEMBL31493128 | 0.83 | HPGD (0.53) | TSHRHTTALOX15CYP3A4ALDH1A1 | |
| SCHEMBL18288014 | 0.83 | HPGD (0.53) | TSHRHTTALOX15CYP3A4ALDH1A1 | |
| SCHEMBL9117716 | 0.83 | ALOX15 (0.46) | TSHRALOX15CYP1A2CYP3A4CYP2C9 | |
| SCHEMBL18288083 | 0.82 | HPGD (0.53) | TSHRMAPK1ALOX15CYP1A2CYP3A4 | |
| SCHEMBL15774869 | 0.80 | TSHR (0.53) | TSHRAPOBEC3AHTTAPOBEC3GMAPK1 | |
| SCHEMBL18288093 | 0.78 | TUBB4A (0.63) | TSHRHTTMAPK1CYP1A2CYP3A4 | |
| SCHEMBL18639610 | 0.78 | MAPT (0.46) | MAPK1ALOX15CYP1A2CYP3A4CYP2C19 |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 182 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| EP-1352083-B2 | COMPOSITIONS AND METHODS FOR DETECTING TARGET MICROORGANISMS IN A SAMPLE | BIOCONTROL SYSTEMS INC (US) | 2013-12-25 | — | — | EP | claimed |
| EP-1500707-B1 | METHOD OF MEASURING NEPRILYSIN ACTIVITY | TAKEDA PHARMACEUTICAL (JP) | 2010-09-15 | — | — | EP | claimed |
| US-7572574-B2 | Method of measuring neprilysin activity | RIKEN (JP) | 2009-08-11 | — | — | US | claimed |
| US-20060008842-A1 | Method of measuring neprilysin activity | TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) | 2006-01-12 | — | — | US | claimed |
| EP-1352083-B1 | COMPOSITIONS AND METHODS FOR DETECTING TARGET MICROORGANISMS IN A SAMPLE | BIOCONTROL SYSTEMS INC (US) | 2005-10-26 | — | — | EP | claimed |
| EP-0946746-B1 | METHOD AND MEDIA FOR THE DETECTION OF YEASTS AND/OR MOLDS IN A SAMPLE | BIOCONTROL SYSTEMS INC (US) | 2005-03-02 | — | — | EP | claimed |
| EP-1500707-A1 | METHOD OF MEASURING NEPRILYSIN ACTIVITY | Riken (JP) | 2005-01-26 | — | — | EP | claimed |
| EP-1156105-B1 | ALPHA-GLYCATED AMINO ACID RELEASING ENZYME | ARKRAY INC (JP) | 2004-09-01 | — | — | EP | claimed |
| EP-1352083-A2 | COMPOSITIONS AND METHODS FOR DETECTING TARGET MICROORGANISMS IN A SAMPLE | BioControl Systems, Inc. (US) | 2003-10-15 | — | — | EP | claimed |
| US-20020058298-A1 | Compositions and methods for detecting target microorganisms in a sample | BIOCONTROL SYSTEM, INC. (US) | 2002-05-16 | — | — | US | claimed |
| EP-1156105-A1 | NOVEL ENZYME | ARKRAY, Inc. (JP) | 2001-11-21 | — | — | EP | claimed |
| US-6022698-A | Method and components for the detection of yeasts and/or molds in a sample | IDEXX LABORATORIES, INCORPORATED (US) | 2000-02-08 | — | — | US | claimed |
| US-5962216-A | MARKER OR ANTICARCINOGENIC/ANTIINFLAMMATORY/ANTITUMOR AGENT LINKED BY CLEAVABLE SEQUENCE TO STABILIZER OF BETA-ALANINE OR SUCCINIC ACID; TARGETED DELIVERY TO CELL, CLEAVAGE BY CELL SPECIFIC FACTOR FOR ENTRY INTO CELL OR EXPRESSION OF MARKER | LA REGION WALLONNE (BE) | 1999-10-05 | — | — | US | claimed |
| US-5854011-A | Method and components for the detection of yeasts and/or molds in a sample | IDEXX LABORATORIES INCORPORATED (US) | 1998-12-29 | — | — | US | claimed |
| EP-0769967-A1 | COMPOUNDS, PHARMACEUTICAL COMPOSITION AND DIAGNOSTIC DEVICE COMPRISING SAME AND THEIR USE | UNIVERSITE CATHOLIQUE DE LOUVAIN (BE) | 1997-05-02 | — | — | EP | claimed |
| WO-1996020949-A1 | PEPTIDE AND PEPTIDE ANALOG PROTEASE INHIBITORS | SIBIA NEUROSCIENCES, INC. (US) | 1996-07-11 | — | — | WO | claimed |
| WO-1996020725-A2 | PEPTIDE, PEPTIDE ANALOG AND AMINO ACID ANALOG PROTEASE INHIBITORS | SIBIA NEUROSCIENCES, INC. (US) | 1996-07-11 | — | — | WO | claimed |
| WO-1996005863-A1 | COMPOUNDS, PHARMACEUTICAL COMPOSITION AND DIAGNOSTIC DEVICE COMPRISING SAME AND THEIR USE | LA REGION WALLONNE (BE) | 1996-02-29 | — | — | WO | claimed |
| US-4335204-A | Easily split substrates for the quantification of proteases | KABI AB (SE) | 1982-06-15 | — | — | US | claimed |
| US-4279810-A | Easily split substrates for the quantification of proteases | KABI AB (SE) | 1981-07-21 | — | — | US | claimed |