SCHEMBL5359996

SCHEMBL5359996

Cc1c(-c2ccc(C#N)cc2)cc(CO)n1Cc1cn[nH]c1C(C)(C)O

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AR P10275 5/20 0.39
CYP11B2 P19099 6/20 0.37
CYP11B1 P15538 4/20 0.34
RIPK3 Q9Y572 1/20 0.34
SLC22A12 Q96S37 3/20 0.33
FNTA P49354 1/20 0.33
FNTB P49356 1/20 0.33
PGGT1B P53609 1/20 0.33
KDM1A O60341 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13362172 0.90 CYP11B2 (0.39) ARCYP11B2RIPK3SLC22A12KDM1A
SCHEMBL5487110 0.81 KMT2A (0.40) ARCYP11B2FNTAFNTB
SCHEMBL5364131 0.78 CYP11B2 (0.40) ARCYP11B2RIPK3KDM1A
SCHEMBL13335446 0.73 AR (0.34) AR
SCHEMBL5366156 0.73 AR (0.37) ARCYP11B2CYP11B1
SCHEMBL5357688 0.69 CYP11B2 (0.36) ARCYP11B2FNTAFNTBPGGT1B
SCHEMBL5353839 0.68 KMT2A (0.39) ARCYP11B2CYP11B1
SCHEMBL5365214 0.68 CYP11B2 (0.43) ARCYP11B2CYP11B1
SCHEMBL5361462 0.66 CYP11B2 (0.41) ARCYP11B2CYP11B1KDM1A
SCHEMBL4919245 0.66 AR (0.69) ARCYP11B2CYP11B1FNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed