SCHEMBL5487110

SCHEMBL5487110

CCOC(=O)c1[nH]ncc1Cn1c(CO)cc(-c2ccc(C#N)cc2)c1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.40
ALDH1A1 P00352 3/20 0.39
MEN1 O00255 2/20 0.39
GAA P10253 2/20 0.39
LMNA P02545 3/20 0.38
MAPT P10636 3/20 0.38
TDP1 Q9NUW8 1/20 0.38
CYP11B2 P19099 1/20 0.37
TSHR P16473 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
AR P10275 3/20 0.37
ELANE P08246 1/20 0.36
SLC34A1 Q06495 1/20 0.36
FNTA P49354 3/20 0.36
FNTB P49356 3/20 0.36
KDM4E B2RXH2 1/20 0.35
HPGD P15428 1/20 0.35
TP53 P04637 1/20 0.35
HRH2 P25021 1/20 0.35
HRH1 P35367 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5353839 0.87 KMT2A (0.39) KMT2AALDH1A1MEN1GAALMNA
SCHEMBL5359996 0.81 AR (0.39) CYP11B2ARFNTAFNTB
SCHEMBL3081244 0.77 ALDH1A1 (0.42) KMT2AALDH1A1MEN1GAALMNA
SCHEMBL5365877 0.74 ELANE (0.40) KMT2AALDH1A1MEN1GAALMNA
SCHEMBL4917896 0.71 AR (0.49) ALDH1A1GAALMNAMAPTTDP1
SCHEMBL13362172 0.71 CYP11B2 (0.39) KMT2AMEN1LMNAMAPTCYP11B2
SCHEMBL14347747 0.70 MAPT (0.39) KMT2AALDH1A1MEN1GAALMNA
SCHEMBL20640817 0.70 ALDH1A1 (0.51) KMT2AALDH1A1MEN1GAALMNA
SCHEMBL5366156 0.68 AR (0.37) CYP11B2AR
SCHEMBL3074166 0.68 AR (0.39) KMT2AALDH1A1MEN1GAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed