SCHEMBL5366156

SCHEMBL5366156

Cc1c(-c2ccc(C#N)cc2)cc(CO)n1Cc1cc(C(F)(F)F)n[nH]1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AR P10275 5/20 0.37
CYP11B2 P19099 4/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.34
GYS1 P13807 1/20 0.34
CCNC P24863 1/20 0.34
CDK8 P49336 1/20 0.34
NSD2 O96028 1/20 0.33
SDHB P21912 1/20 0.33
CYP11B1 P15538 1/20 0.32
CNR1 P21554 1/20 0.32
KIF11 P52732 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5357164 0.89 CYP11B2 (0.39) ARCYP11B2PTGDR2GYS1CCNC
SCHEMBL5362074 0.84 CYP11B2 (0.35) ARCYP11B2PTGDR2GYS1CCNC
SCHEMBL5357234 0.84 CYP11B2 (0.37) ARCYP11B2PTGDR2GYS1CCNC
SCHEMBL5353540 0.81 CYP11B2 (0.38) ARCYP11B2PTGDR2GYS1CCNC
SCHEMBL5367787 0.78 CYP11B2 (0.35) CYP11B2PTGDR2GYS1CCNCCDK8
SCHEMBL5354656 0.75 AR (0.40) ARCYP11B2CCNCCDK8
SCHEMBL5355359 0.74 CYP11B2 (0.37) ARCYP11B2NSD2CYP11B1
SCHEMBL5359725 0.74 AR (0.48) ARPTGDR2GYS1SDHB
SCHEMBL5358762 0.73 CYP11B2 (0.40) ARCYP11B2CCNCCDK8
SCHEMBL5359996 0.73 AR (0.39) ARCYP11B2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed
WO-2007145349-A2 SUBSTITUTED PYRROLE DERIVATIVES TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-12-21 WO disclosed