SCHEMBL536111

SCHEMBL536111

O=C(O)c1cccc2nc(-c3ccc(-c4ccccc4F)c(F)c3)[nH]c12

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 14/20 0.59
HDAC6 Q9UBN7 2/20 0.47
KDM4E B2RXH2 2/20 0.46
RAB9A P51151 2/20 0.46
TP53 P04637 1/20 0.46
MAPT P10636 1/20 0.46
ACMSD Q8TDX5 1/20 0.44
NPC1 O15118 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL505378 0.93 DHODH (0.69) DHODHHDAC6KDM4ERAB9AACMSD
SCHEMBL506154 0.90 DHODH (0.67) DHODHHDAC6KDM4ERAB9AACMSD
SCHEMBL505457 0.88 DHODH (0.68) DHODHHDAC6KDM4ERAB9A
SCHEMBL6840296 0.87 RAB9A (0.56) DHODHKDM4ERAB9ANPC1ALDH1A1
SCHEMBL536117 0.86 DHODH (0.60) DHODHHDAC6
SCHEMBL505990 0.85 DHODH (0.57) DHODHHDAC6KDM4EACMSDALDH1A1
SCHEMBL536113 0.84 DHODH (0.58) DHODHHDAC6KDM4ERAB9AALDH1A1
SCHEMBL505906 0.84 DHODH (0.58) DHODHHDAC6KDM4ERAB9AACMSD
SCHEMBL505582 0.84 DHODH (0.64) DHODHKDM4ETP53MAPTALDH1A1
SCHEMBL6840189 0.81 PIN1 (0.58) DHODHKDM4ERAB9ATP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414328-A2 DIHYDROOROTATE DEHYDROGENASE INHIBITORS Merck Serono S.A. (CH) 2012-02-08 EP disclosed