SCHEMBL536398

SCHEMBL536398

Oc1ccccc1N1Nc2ccccc2N1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.41
GAA P10253 4/20 0.41
MAPT P10636 2/20 0.41
POLB P06746 2/20 0.41
XBP1 P17861 1/20 0.41
MAPK1 P28482 1/20 0.41
ALDH1A1 P00352 3/20 0.39
HPGD P15428 2/20 0.39
HIF1A Q16665 2/20 0.39
HSD17B10 Q99714 2/20 0.39
CA2 P00918 2/20 0.39
CA4 P22748 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
LMNA P02545 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
ALOX15 P16050 2/20 0.39
NPC1 O15118 1/20 0.39
CA12 O43570 1/20 0.39
GMNN O75496 1/20 0.39
EGFR P00533 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28402822 0.77 LMNA (0.51) KDM4EGAAMAPTPOLBALDH1A1
SCHEMBL31410938 0.75 TRPM4 (0.36) KDM4EGAAMAPTPOLBMAPK1
SCHEMBL27436605 0.71 KDM4E (0.36) KDM4EGAAMAPTPOLBXBP1
SCHEMBL14429576 0.70 IDO1 (0.37) KDM4EGAAMAPTPOLBXBP1
SCHEMBL15065849 0.69 MEN1 (0.36) KDM4EGAAMAPTPOLBXBP1
SCHEMBL8541096 0.68 KDM4E (0.37) KDM4EGAAMAPTPOLBXBP1
SCHEMBL28719531 0.68 ALOX5 (0.33) KDM4EGAAMAPTALDH1A1SMN1; SMN2
SCHEMBL13879920 0.67 LMNA (0.37) KDM4EGAAMAPTPOLBALDH1A1
SCHEMBL22702465 0.67 KDM4E (0.33) KDM4EGAAMAPTPOLBXBP1
SCHEMBL8979742 0.65 GAA (0.37) KDM4EGAAHPGDSMN1; SMN2ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 61 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4251696-B1 UV RESISTANT SMMA COPOLYMERS WITH LOW HAZE AND HIGH CLARITY INEOS STYROLUTION GROUP GMBH (DE) 2024-11-20 EP claimed
CN-117165127-A Sealing material for hydrogen production electrolytic tank and gasket structure thereof 镇江春环密封件集团有限公司 2023-12-05 CN claimed
EP-1926770-B1 COLOR FAST POLYURETHANES CIBA HOLDING INC (CH) 2013-06-19 EP claimed
EP-0236413-B1 SUNGLASS LENSES TANOPTIC AG (CH) 1994-06-08 EP claimed
EP-0363318-B1 Process for the preparation of benzotriazole derivatives CIBA GEIGY AG (CH) 1994-03-02 EP claimed
EP-0419412-B1 Process for the preparation of benzotriazoles CIBA GEIGY AG (CH) 1993-11-10 EP claimed
EP-0303986-B1 MULTIPURPOSE POLYMER BOUND STABILIZERS ATOCHEM NORTH AMERICA, INC. (US) 1992-07-29 EP claimed
EP-0419412-A2 Process for the preparation of benzotriazoles CIBA-GEIGY AG (CH) 1991-03-27 EP claimed
EP-0363318-A1 Process for the preparation of benzotriazole derivatives CIBA-GEIGY AG (CH) 1990-04-11 EP claimed
EP-0099231-B1 POLYPHENYLENE ETHER RESIN COMPOSITION MITSUBISHI GAS CHEMICAL COMPANY, INC. (JP) 1987-11-25 EP claimed
EP-0045040-B1 POWDER COATING COMPOSITION FOR AUTOMOTIVE TOPCOAT AND THE COATED ARTICLE E.I. DU PONT DE NEMOURS AND COMPANY (US) 1984-10-24 EP claimed
EP-4305098-A1 USE OF AT LEAST ONE SULFUR-CONTAINING AMINO ACID FOR STABILIZING RECYCLED THERMOPLASTICS, STABILIZED RECYCLED THERMOPLASTIC, STABILIZER COMPOSITION, MASTERBATCH, AND MOLDING COMPOUND OR MOLDED PART Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2024-01-17 EP disclosed
CN-117165127-A Sealing material for hydrogen production electrolytic tank and gasket structure thereof 镇江春环密封件集团有限公司 2023-12-05 CN disclosed
WO-2022243354-A1 USE OF AT LEAST ONE SULFUR-CONTAINING AMINO ACID FOR STABILIZING RECYCLED THERMOPLASTICS, STABILIZED RECYCLED THERMOPLASTIC, STABILIZER COMPOSITION, MASTERBATCH, AND MOLDING COMPOUND OR MOLDED PART Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2022-11-24 WO disclosed
EP-4069757-A1 FLAME RETARDANT POLYMER COMPRISING PHOSPHORUS-CONTAINING REPEATING UNITS, PLASTIC COMPOSITION COMPRISING THE FLAME RETARDANT POLYMER, PROCESS FOR PRODUCING THE FLAME RETARDANT POLYMER AND USE THEREOF Fraunhofer-Gesellschaft zur Förderung der angewandten Forschung e.V. (DE) 2022-10-12 EP disclosed
EP-0323408-A1 2-(2-Hydroxyphenyl)-benztriazole derivatives CIBA-GEIGY AG (CH) 1989-07-05 EP disclosed
EP-0180548-B1 COATINGS STABILIZED AGAINST THE ACTION OF LIGHT CIBA-GEIGY AG (CH) 1989-06-28 EP disclosed
EP-0181283-B1 ISOMERIC MIXTURES OF METAL SALICYLATES, THEIR PREPARATION AND UTILISATION CIBA-GEIGY AG (CH) 1988-09-28 EP disclosed
EP-0109930-B1 CHROMOGENIC BIS-QUINAZOLINE COMPOUNDS, METHOD OF PREPARING THEM AND THEIR USE AS CHROMOGENES IN PRESSURE-SENSITIVE OR HEAT-SENSITIVE RECORDING MATERIALS CIBA-GEIGY AG (CH) 1986-09-17 EP disclosed
EP-0180548-A2 Coatings stabilized against the action of light CIBA-GEIGY AG (CH) 1986-05-07 EP disclosed