Disulfiram

Disulfiram

SCHEMBL5364281

CCN(CC)C(=S)SSC(=S)N(CC)CC.[Hg]

nearest known ligand 0.94

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ALDH2

The experimentally established mechanism targets of Disulfiram. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH2 known ✓ P05091 7/20 0.94
ALDH1A1 P00352 10/20 0.94
MGLL Q99685 7/20 0.94
EHMT2 Q96KQ7 4/20 0.94
EHMT1 Q9H9B1 4/20 0.94
PHGDH O43175 3/20 0.94
CYP3A4 P08684 3/20 0.94
HTT P42858 3/20 0.94
ABCB11 O95342 2/20 0.94
GSDMD P57764 2/20 0.94
LMNA P02545 2/20 0.94
TP53 P04637 2/20 0.94
HSP90AA1 P07900 2/20 0.94
FBP1 P09467 2/20 0.94
MAPT P10636 2/20 0.94
PKM P14618 2/20 0.94
HPGD P15428 2/20 0.94
ALOX15 P16050 2/20 0.94
ALOX12 P18054 2/20 0.94
LOX P28300 2/20 0.94

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Disulfiram SCHEMBL4654748 0.97 ALDH1A1 (1.00) ALDH1A1ALDH2MGLLEHMT2EHMT1
Disulfiram SCHEMBL27213 0.97 ALDH1A1 (1.00) ALDH1A1ALDH2MGLLEHMT2EHMT1
Disulfiram SCHEMBL5961375 0.94 ALDH1A1 (0.94) ALDH1A1ALDH2MGLLEHMT2EHMT1
Disulfiram SCHEMBL29067672 0.94 ALDH1A1 (0.94) ALDH1A1ALDH2MGLLEHMT2EHMT1
Disulfiram SCHEMBL28246322 0.94 ALDH1A1 (0.94) ALDH1A1ALDH2MGLLEHMT2EHMT1
Disulfiram SCHEMBL28867973 0.94 ALDH1A1 (0.94) ALDH1A1ALDH2MGLLEHMT2EHMT1
Disulfiram SCHEMBL10886601 0.94 ALDH1A1 (0.94) ALDH1A1ALDH2MGLLEHMT2EHMT1
Disulfiram SCHEMBL11155542 0.94 ALDH1A1 (0.94) ALDH1A1ALDH2MGLLEHMT2EHMT1
Disulfiram SCHEMBL31719635 0.94 ALDH1A1 (0.94) ALDH1A1ALDH2MGLLEHMT2EHMT1
Disulfiram SCHEMBL28998625 0.94 ALDH1A1 (0.94) ALDH1A1ALDH2MGLLEHMT2EHMT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7252957-B2 Identification of etiology of autism IMMUNOSCIENCES LAB., INC. (US) 2007-08-07 US disclosed
US-20050170333-A1 Identification of etiology of autism Knobbe, Martens, Olson & Bear, LLP 2005-08-04 US disclosed