SCHEMBL5364936

SCHEMBL5364936

Cc1cc(=O)[nH]nc1Cc1ccc(Cl)c(Oc2cccc(C#N)c2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRMT5 O14744 1/20 0.40
WDR77 Q9BQA1 1/20 0.40
P2RX3 P56373 4/20 0.39
DRD4 P21917 1/20 0.39
FNTA P49354 1/20 0.39
FNTB P49356 1/20 0.39
PGGT1B P53609 1/20 0.39
CYP3A4 P08684 3/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
KCNH2 Q12809 3/20 0.37
HTR2A P28223 2/20 0.37
SLC6A4 P31645 1/20 0.37
EPAS1 Q99814 3/20 0.36
NR1H4 Q96RI1 1/20 0.35
EGFR P00533 1/20 0.35
ERBB2 P04626 1/20 0.35
ERBB3 P21860 1/20 0.35
ERBB4 Q15303 1/20 0.35
AR P10275 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5377272 0.87 PRMT5 (0.43) PRMT5WDR77P2RX3DRD4FNTA
SCHEMBL5373462 0.87 CYP3A4 (0.41) PRMT5WDR77P2RX3CYP3A4CYP2C9
SCHEMBL5364878 0.86 PARP1 (0.43) FNTAFNTBPGGT1BCYP3A4CYP2C9
SCHEMBL5377579 0.84 CYP3A4 (0.52) PRMT5WDR77P2RX3DRD4FNTA
SCHEMBL14570769 0.83 CYP3A4 (0.53) PRMT5WDR77P2RX3DRD4FNTA
SCHEMBL5377601 0.82 PARP1 (0.38) CYP3A4CYP2C9CYP2C19KCNH2TSHR
SCHEMBL4370994 0.81 P2RX3 (0.41) PRMT5WDR77P2RX3DRD4FNTA
SCHEMBL4808827 0.80 CYP3A4 (0.48) PRMT5WDR77P2RX3DRD4FNTA
SCHEMBL5368822 0.79 PARP1 (0.33) P2RX3CYP3A4CYP2C9CYP2C19TSHR
SCHEMBL5370838 0.78 CYP3A4 (0.45) CYP3A4CYP2C9CYP2C19KCNH2EPAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed