SCHEMBL5377601

SCHEMBL5377601

Cc1cc(=O)[nH]nc1Cc1ccc(Cl)c(Oc2cc(Cl)cc(Cl)c2)c1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 12/20 0.38
CYP3A4 P08684 3/20 0.37
CYP2C9 P11712 1/20 0.37
TSHR P16473 1/20 0.37
CYP2C19 P33261 1/20 0.37
CCNE2 O96020 2/20 0.34
CDK4 P11802 2/20 0.34
CCND1 P24385 2/20 0.34
CCNE1 P24864 2/20 0.34
CDK2 P24941 2/20 0.34
KCNH2 Q12809 1/20 0.33
LMNA P02545 1/20 0.33
ADORA2A P29274 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5373462 0.89 CYP3A4 (0.41) PARP1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL5364878 0.84 PARP1 (0.43) PARP1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL5364936 0.82 PRMT5 (0.40) CYP3A4CYP2C9TSHRCYP2C19KCNH2
SCHEMBL5368714 0.80 CYP3A4 (0.53) PARP1CYP3A4
SCHEMBL5375026 0.80 CYP3A4 (0.46) PARP1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL5373600 0.78 CYP3A4 (0.45) PARP1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL5368822 0.77 PARP1 (0.33) PARP1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL4805650 0.76 CYP3A4 (0.47) CYP3A4CCNE2CDK4CCND1CCNE1
SCHEMBL5367070 0.73 CYP3A4 (0.37) PARP1CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL5374044 0.72 PARP1 (0.41) PARP1CYP3A4CYP2C9TSHRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed