SCHEMBL5365201

SCHEMBL5365201

CN(CCOC(N)=O)c1cc(Cc2ccc(Cl)c(Oc3cccc(Cl)c3)c2)n[nH]c1=O

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.40
ICAM1 P05362 1/20 0.35
SELE P16581 1/20 0.35
VCAM1 P19320 1/20 0.35
KDM4E B2RXH2 2/20 0.33
PARP1 P09874 5/20 0.33
PRMT5 O14744 1/20 0.33
WDR77 Q9BQA1 1/20 0.33
DAO P14920 2/20 0.33
SLC6A4 P31645 2/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A3 Q01959 1/20 0.32
HTR2A P28223 1/20 0.32
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31
P2RX4 Q99571 2/20 0.31
FAAH O00519 1/20 0.31
MGLL Q99685 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5368522 0.88 CYP3A4 (0.43) CYP3A4KDM4EPARP1PRMT5WDR77
SCHEMBL5368691 0.76 CYP3A4 (0.47) CYP3A4PARP1PRMT5WDR77DAO
SCHEMBL5375576 0.76 PARP1 (0.39) CYP3A4PARP1DAOSLC6A4HTR2A
SCHEMBL14559738 0.75 THRA (0.31) CYP3A4PARP1DAO
SCHEMBL5377396 0.74 CYP3A4 (0.41) CYP3A4PRMT5WDR77SLC6A4HTR2A
SCHEMBL5365181 0.73 CYP3A4 (0.67) CYP3A4PRMT5WDR77SLC6A4SLC6A2
SCHEMBL5370255 0.70 CYP3A4 (0.45) CYP3A4KDM4EPARP1SLC6A4FAAH
SCHEMBL4805444 0.69 CYP3A4 (0.45) CYP3A4SLC6A4SLC6A2SLC6A3HTR2A
SCHEMBL5374033 0.69 CYP3A4 (0.41) CYP3A4PARP1PRMT5WDR77SLC6A4
SCHEMBL5385763 0.69 CYP3A4 (0.43) CYP3A4PARP1PRMT5WDR77DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed