SCHEMBL5368522

SCHEMBL5368522

CN(CCO)c1cc(Cc2ccc(Cl)c(Oc3cccc(Cl)c3)c2)n[nH]c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.43
SLC6A4 P31645 2/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A3 Q01959 1/20 0.35
RHEB Q15382 2/20 0.34
PRMT5 O14744 1/20 0.34
WDR77 Q9BQA1 1/20 0.34
DAO P14920 2/20 0.33
KCNH2 Q12809 2/20 0.33
HTR2A P28223 1/20 0.33
PARP1 P09874 3/20 0.33
STK4 Q13043 1/20 0.33
STK3 Q13188 1/20 0.33
LRRK2 Q5S007 1/20 0.33
KDM4E B2RXH2 2/20 0.32
TRPC5 Q9UL62 3/20 0.32
TRPC4 Q9UBN4 1/20 0.32
FNTA P49354 1/20 0.32
FNTB P49356 1/20 0.32
PGGT1B P53609 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5365201 0.88 CYP3A4 (0.40) CYP3A4SLC6A4SLC6A2SLC6A3PRMT5
SCHEMBL14559738 0.86 THRA (0.31) CYP3A4DAOPARP1
SCHEMBL5368691 0.80 CYP3A4 (0.47) CYP3A4SLC6A4SLC6A2SLC6A3PRMT5
SCHEMBL5375576 0.80 PARP1 (0.39) CYP3A4SLC6A4DAOKCNH2HTR2A
SCHEMBL5377396 0.78 CYP3A4 (0.41) CYP3A4SLC6A4PRMT5WDR77KCNH2
SCHEMBL5365181 0.77 CYP3A4 (0.67) CYP3A4SLC6A4SLC6A2SLC6A3RHEB
SCHEMBL5373478 0.74 CYP3A4 (0.38) CYP3A4SLC6A4DAOKCNH2HTR2A
SCHEMBL5370255 0.73 CYP3A4 (0.45) CYP3A4SLC6A4PARP1KDM4EFAAH
SCHEMBL5374033 0.72 CYP3A4 (0.41) CYP3A4SLC6A4PRMT5WDR77KCNH2
SCHEMBL5385763 0.72 CYP3A4 (0.43) CYP3A4PRMT5WDR77DAOPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed