SCHEMBL5374482

SCHEMBL5374482

O=c1ccc(Cc2ccc(C(F)(F)F)c(Oc3cccc(Cl)c3)c2)n[nH]1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.61
EPAS1 Q99814 1/20 0.46
AR P10275 1/20 0.40
PTGS1 P23219 1/20 0.35
P2RX4 Q99571 2/20 0.35
HTR2A P28223 2/20 0.35
SLC6A4 P31645 2/20 0.35
KCNH2 Q12809 2/20 0.35
KDR P35968 1/20 0.35
AKR1B1 P15121 2/20 0.34
FABP4 P15090 1/20 0.34
FNTA P49354 1/20 0.33
FNTB P49356 1/20 0.33
PGGT1B P53609 1/20 0.33
MAPK10 P53779 1/20 0.33
AHR P35869 1/20 0.33
ICAM1 P05362 1/20 0.33
SELE P16581 1/20 0.33
VCAM1 P19320 1/20 0.33
PRMT5 O14744 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5377568 0.89 CYP3A4 (0.47) CYP3A4ARHTR2ASLC6A4KCNH2
SCHEMBL5366909 0.88 CYP3A4 (0.46) CYP3A4KDRAKR1B1
SCHEMBL5377723 0.87 CYP3A4 (0.66) CYP3A4EPAS1P2RX4HTR2ASLC6A4
SCHEMBL5365181 0.86 CYP3A4 (0.67) CYP3A4HTR2ASLC6A4KCNH2AKR1B1
SCHEMBL5373732 0.85 CYP3A4 (0.45) CYP3A4EPAS1ARKCNH2FNTA
SCHEMBL5373755 0.85 CYP3A4 (0.45) CYP3A4EPAS1ARPTGS1P2RX4
SCHEMBL5368939 0.84 CYP3A4 (0.64) CYP3A4PTGS1P2RX4HTR2ASLC6A4
SCHEMBL5377627 0.84 CYP3A4 (0.64) CYP3A4P2RX4HTR2ASLC6A4KCNH2
SCHEMBL5374946 0.83 CYP3A4 (0.42) CYP3A4ARKDRAKR1B1PRMT5
SCHEMBL5370245 0.83 CYP3A4 (0.63) CYP3A4PTGS1HTR2ASLC6A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed
US-7189718-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-03-13 US disclosed