SCHEMBL5366188

SCHEMBL5366188

O=C(NC(C(=O)C1CC1c1ccccc1)C1CCNCC1)c1ccc(O)cc1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DEGS1 O15121 2/20 0.44
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
MAPK1 P28482 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
KDM1A O60341 5/20 0.39
MAOB P27338 4/20 0.39
MAOA P21397 3/20 0.39
HDAC4 P56524 1/20 0.39
SMYD3 Q9H7B4 2/20 0.38
CDK2 P24941 1/20 0.38
AKT1 P31749 1/20 0.38
HPGD P15428 1/20 0.38
EPHX2 P34913 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5368190 0.89 EPHX2 (0.52) ALDH1A1KDM1AMAOBMAOAEPHX2
SCHEMBL5362652 0.82 AKT1 (0.41) ALDH1A1SMYD3CDK2AKT1
SCHEMBL5353674 0.77 KDM1A (0.45) ALDH1A1MAPTMAPK1TDP1KDM1A
SCHEMBL5360331 0.77 SCN3A (0.39) DEGS1KDM1AMAOBMAOASMYD3
SCHEMBL5362924 0.77 KMT2A (0.41) ALDH1A1KDM4ETDP1SMYD3CDK2
SCHEMBL5371022 0.76 KMT2A (0.49) KDM4EMAPTSMYD3CDK2AKT1
SCHEMBL5367918 0.76 ALDH1A1 (0.41) ALDH1A1MAPTKDM1ASMYD3CDK2
SCHEMBL5364811 0.73 MEN1 (0.42) ALDH1A1KDM4ESMYD3CDK2AKT1
SCHEMBL5371067 0.71 NPC1 (0.42) SMYD3CDK2AKT1
SCHEMBL5366087 0.71 HPGD (0.44) ALDH1A1MAPTSMYD3HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7259157-B2 N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists MERCK & CO., INC. (US) 2007-08-21 US disclosed